SCHEMBL10285249

SCHEMBL10285249

CN(C(=O)OC(C)(C)C)C1CCN(CCn2c(=O)cnc3ccc(C#N)cc32)CC1

nearest known ligand 0.51

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 14/20 0.51
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
EGLN1 Q9GZT9 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL708597 0.84 KCNH2 (0.51) KCNH2CYP3A4CYP2D6
SCHEMBL12002207 0.84 KCNH2 (0.54) KCNH2
SCHEMBL706674 0.79 KCNH2 (0.45) KCNH2CYP3A4CYP2D6EGLN1
SCHEMBL708368 0.78 KCNH2 (0.56) KCNH2CYP3A4CYP2D6
SCHEMBL14679203 0.77 KCNH2 (0.56) KCNH2CYP3A4CYP2D6
SCHEMBL14610965 0.77 CDK8 (0.42) KCNH2EGLN1
SCHEMBL922035 0.77 KCNH2 (0.57) KCNH2CYP3A4CYP2D6
SCHEMBL12002208 0.76 KCNH2 (0.55) KCNH2CYP3A4CYP2D6
SCHEMBL19094697 0.76 KCNH2 (0.49) KCNH2
SCHEMBL2797848 0.75 KCNH2 (0.56) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2468743-A1 Nitrogen-containing bicyclic compounds useful as antibacterial agents Toyama Chemical Co., Ltd. (JP) 2012-06-27 EP disclosed
EP-1900732-A1 NOVEL NITROGENATED HETEROCYCLIC COMPOUND AND SALT THEREOF TOYAMA CHEMICAL CO., LTD. (JP) 2008-03-19 EP disclosed