SCHEMBL10286248

SCHEMBL10286248

Cc1nnc2n1-c1cnc(-c3ccncc3-c3ccccc3)nc1N1CCOCC21

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MTOR P42345 8/20 0.39
PIK3CA P42336 3/20 0.36
GAA P10253 1/20 0.35
TRPM8 Q7Z2W7 1/20 0.35
NUDT1 P36639 1/20 0.34
ATR Q13535 5/20 0.34
LMNA P02545 2/20 0.34
HTT P42858 1/20 0.34
ATRIP Q8WXE1 1/20 0.33
OXTR P30559 1/20 0.33
AVPR1A P37288 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1288867 0.89 MTOR (0.35) MTORPIK3CAGAATRPM8NUDT1
SCHEMBL1688527 0.83 MTOR (0.35) MTORPIK3CATRPM8NUDT1ATR
SCHEMBL1688532 0.76 GAA (0.34) MTORGAATRPM8LMNAHTT
SCHEMBL1288910 0.76 MTOR (0.35) MTORPIK3CAGAATRPM8NUDT1
SCHEMBL2688281 0.76 GAA (0.34) MTORGAATRPM8LMNAHTT
SCHEMBL2689714 0.75 MTOR (0.37) MTORPIK3CAATRATRIP
SCHEMBL1288812 0.75 PLK1 (0.41)
SCHEMBL1288808 0.75 PLK1 (0.41)
SCHEMBL1288520 0.74 PLK1 (0.42)
SCHEMBL1288526 0.74 PLK1 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012048129-A2 INHIBITORS OF POLO-LIKE KINASE ELAN PHARMACEUTICALS, INC. (US) 2012-04-12 WO disclosed