SCHEMBL1029494

SCHEMBL1029494

CC(=O)N1C/C(=C\c2ccc(F)cc2)c2c(c(C(=O)N(C(C)=O)N3CC4CCCC4C3)nn2-c2ccc(Cl)cc2)C1

nearest known ligand 0.48

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 19/20 0.48
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
TP53 P04637 1/20 0.40
HPGD P15428 1/20 0.40
CNR2 P34972 8/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1029496 1.00 CNR1 (0.48) CNR1KDM4EALDH1A1TP53HPGD
SCHEMBL1028799 0.85 CNR1 (0.52) CNR1CNR2
SCHEMBL5318133 0.82 CNR1 (0.56) CNR1KDM4EALDH1A1TP53HPGD
SCHEMBL5318134 0.82 CNR1 (0.56) CNR1KDM4EALDH1A1TP53HPGD
SCHEMBL1029218 0.80 CNR1 (0.51) CNR1KDM4EALDH1A1TP53HPGD
SCHEMBL1029217 0.80 CNR1 (0.51) CNR1KDM4EALDH1A1TP53HPGD
SCHEMBL1030628 0.79 CNR1 (0.52) CNR1CNR2
SCHEMBL1030626 0.79 CNR1 (0.52) CNR1CNR2
SCHEMBL1029770 0.77 CNR1 (0.54) CNR1CNR2
SCHEMBL1029771 0.77 CNR1 (0.54) CNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1804791-B1 TETRAHYDRO PYRIDINYL PYRAZOLE CANNABINOID MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2011-01-19 EP disclosed