SCHEMBL10312162

SCHEMBL10312162

CP(C)(=O)c1ccc(Nc2nc(/C=C/c3cccc(Cl)c3)nc(Nc3cc(C4CC4)[nH]n3)n2)cc1

nearest known ligand 0.45

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
IGF1R P08069 16/20 0.45
CCNA2 P20248 1/20 0.43
CDK2 P24941 1/20 0.43
CCNA1 P78396 1/20 0.43
NEK1 Q96PY6 1/20 0.40
ULK1 O75385 1/20 0.40
SRC P12931 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10312087 0.90 IGF1R (0.43) IGF1RNEK1ULK1SRC
SCHEMBL10312178 0.88 CCNA2 (0.45) IGF1RCCNA2CDK2CCNA1NEK1
SCHEMBL10312194 0.87 AURKA (0.41) IGF1RSRC
SCHEMBL10312154 0.82 IGF1R (0.45) IGF1RCCNA2CDK2CCNA1
SCHEMBL10312148 0.79 IGF1R (0.50) IGF1RCCNA2CDK2CCNA1
SCHEMBL10312173 0.78 IGF1R (0.54) IGF1R
SCHEMBL10312132 0.78 NTRK1 (0.47) IGF1R
SCHEMBL10312128 0.78 PAK4 (0.47) IGF1R
SCHEMBL10312196 0.77 HRH4 (0.57) IGF1RSRC
SCHEMBL10312219 0.77 AURKA (0.41) IGF1RSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2440055-B1 STYRYL-TRIAZINE DERIVATIVES AND THEIR THERAPEUTICAL APPLICATIONS CALIFORNIA CAPITAL EQUITY LLC (US) 2015-03-11 EP disclosed
US-20120178758-A1 STYRYL-TRIAZINE DERIVATIVES AND THEIR THERAPEUTICAL APPLICATIONS CALIFORNIA CAPITAL EQUITY, LLC (US) 2012-07-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120178758-A1 STYRYL-TRIAZINE DERIVATIVES AND THEIR THERAPEUTICAL APPLICATIONS STK25, STK35, SGK2 IGF1R 1148/4885CCNA2 1229/4885CDK2 225/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.