SCHEMBL10315902

SCHEMBL10315902

Cc1ccccc1-n1c(O)nnc1-c1cc(C(=O)O)c(O)cc1OCc1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 3/20 0.45
MYC P01106 1/20 0.42
HSP90AA1 P07900 1/20 0.42
HSP90AB1 P08238 1/20 0.42
PTGER1 P34995 8/20 0.41
NOTUM Q6P988 1/20 0.40
RXRA P19793 1/20 0.40
RXRB P28702 1/20 0.40
RXRG P48443 1/20 0.40
MAOB P27338 1/20 0.39
CYP1A2 P05177 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10170480 0.93 MCL1 (0.43) MCL1MYCPTGER1NOTUMRXRA
SCHEMBL10170476 0.92 MCL1 (0.45) MCL1MYCHSP90AA1HSP90AB1PTGER1
SCHEMBL10315951 0.91 KDM4E (0.43) MCL1MYCHSP90AA1HSP90AB1NOTUM
SCHEMBL10170484 0.88 HSP90AA1 (0.58) HSP90AA1HSP90AB1
SCHEMBL10170473 0.86 NOTUM (0.41) MCL1MYCHSP90AA1HSP90AB1PTGER1
SCHEMBL3305899 0.85 HSP90AA1 (0.50) HSP90AA1HSP90AB1
SCHEMBL10170472 0.83 KDM4E (0.43) MYCHSP90AA1HSP90AB1NOTUMMAOB
SCHEMBL10170483 0.83 HSP90AA1 (0.52) HSP90AA1HSP90AB1
SCHEMBL645182 0.82 BRD4 (0.39) PTGER1CYP1A2
SCHEMBL3305910 0.80 HSP90AA1 (0.45) HSP90AA1HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2023922-B1 TRIAZOLE DERIVATIVES II MERCK PATENT GMBH (DE) 2012-07-11 EP disclosed
WO-2007134678-A2 TRIAZOLE DERIVATIVES II MERCK PATENT GMBH (DE) 2007-11-29 WO disclosed