SCHEMBL10320848

SCHEMBL10320848

CN1Cc2ccccc2C(=O)c2cc(CC(=O)O)ccc21

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 5/20 0.54
PARK7 Q99497 1/20 0.47
KDM4E B2RXH2 2/20 0.42
ALOX15 P16050 1/20 0.42
TSHR P16473 1/20 0.42
SIRT1 Q96EB6 1/20 0.42
HRH1 P35367 3/20 0.42
ACHE P22303 1/20 0.42
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
HSD17B10 Q99714 1/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11456433 0.90 AKR1B1 (0.57) AKR1B1PARK7KDM4EALOX15TSHR
SCHEMBL11455808 0.89 AKR1B1 (0.42) AKR1B1PARK7KDM4EALOX15TSHR
SCHEMBL11467885 0.87 AKR1B1 (0.40) AKR1B1ACHE
SCHEMBL11467897 0.87 AKR1B1 (0.40) AKR1B1ACHEALDH1A1
SCHEMBL11457263 0.87 TSHR (0.44) AKR1B1TSHRACHEALDH1A1HPGD
SCHEMBL11463851 0.86 AKR1B1 (0.50) AKR1B1PARK7KDM4EALOX15TSHR
SCHEMBL11457865 0.85 AKR1B1 (0.52) AKR1B1PARK7KDM4EALOX15TSHR
SCHEMBL11455791 0.85 MEN1 (0.43) AKR1B1ALDH1A1HPGDHSD17B10
SCHEMBL11464142 0.84 AKR1B1 (0.44) AKR1B1PARK7ALDH1A1PTGDR2
SCHEMBL11474317 0.84 AKR1B1 (0.49) AKR1B1PARK7KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4230703-A ANALGESICS; ANTIINFLAMMATORY AGENTS TEIKOKU HORMONE MFG. CO., LTD. (JP) 1980-10-28 US claimed
WO-2014176460-A1 METHODS OF TREATING BEHAVIORIAL AND/OR MENTAL DISORDERS CHAU DAVID T (US) 2014-10-30 WO disclosed
US-8486922-B2 Composition CHEN CHIEN-HUNG (TW) 2013-07-16 US disclosed
US-20120183600-A1 NOVEL COMPOSITION FOR TREATING METABOLIC SYNDROME AND OTHER CONDITIONS CHEN CHIEN-HUNG (US) 2012-07-19 US disclosed
US-4230703-A ANALGESICS; ANTIINFLAMMATORY AGENTS TEIKOKU HORMONE MFG. CO., LTD. (JP) 1980-10-28 US disclosed