SCHEMBL10328255

SCHEMBL10328255

CCNC(=O)Nc1ccc2ncc(C)nc2n1

nearest known ligand 0.70

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 20/20 0.70
MAPK8 P45983 14/20 0.70
MAPK9 P45984 14/20 0.70
MAPK10 P53779 14/20 0.70
MAPK1 P28482 13/20 0.70
MAPK14 Q16539 1/20 0.70

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5449305 0.86 PIK3CA (0.70) PIK3CAMAPK8MAPK9MAPK10MAPK1
SCHEMBL5441554 0.85 PIK3CA (0.71) PIK3CAMAPK8MAPK9MAPK10MAPK1
SCHEMBL5455686 0.85 PIK3CA (0.71) PIK3CAMAPK8MAPK9MAPK10MAPK1
SCHEMBL10328053 0.84 PIK3CA (0.64) PIK3CAMAPK8MAPK9MAPK10MAPK1
SCHEMBL5454900 0.83 PIK3CA (0.83) PIK3CAMAPK8MAPK9MAPK10MAPK1
SCHEMBL5447520 0.83 PIK3CA (1.00) PIK3CAMAPK8MAPK9MAPK10MAPK1
SCHEMBL14506618 0.83 PIK3CA (1.00) PIK3CAMAPK8MAPK9MAPK10MAPK1
SCHEMBL5622877 0.83 PIK3CA (0.76) PIK3CAMAPK8MAPK9MAPK10MAPK1
SCHEMBL5623757 0.82 PIK3CA (0.83) PIK3CAMAPK8MAPK9MAPK10MAPK1
SCHEMBL10328380 0.82 PIK3CA (0.61) PIK3CAMAPK8MAPK9MAPK10MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1962854-B1 PYRIDOPYRAZINE DERIVATIVES AND USE THEREOF AS MODULATORS OF THE SIGNAL TRANSDUCTION PATHS TERNA ZENTARIS GMBH (DE) 2015-05-06 EP disclosed
US-8217042-B2 Pyridopyrazines and their use as modulators of kinases ZENTARIS GMBH (DE) 2012-07-10 US disclosed
US-8217042-B2 Pyridopyrazines and their use as modulators of kinases ZENTARIS GMBH (DE) 2012-07-10 US disclosed