SCHEMBL10340640

SCHEMBL10340640

CCOC(=O)c1cnn(-c2cccc(CC)c2)c1N

nearest known ligand 0.78

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.78
ALDH1A1 P00352 4/20 0.75
HPGD P15428 3/20 0.75
RAB9A P51151 2/20 0.67
TSHR P16473 3/20 0.66
SMN1; SMN2 Q16637 2/20 0.66
MAPT P10636 5/20 0.60
KMT2A Q03164 2/20 0.59
MEN1 O00255 1/20 0.59
NPC1 O15118 3/20 0.59
TP53 P04637 2/20 0.59
NPSR1 Q6W5P4 1/20 0.53
CYP1A2 P05177 1/20 0.53
CYP2C19 P33261 1/20 0.53
RECQL P46063 1/20 0.53
LMNA P02545 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16479382 0.92 HTT (0.73) HTTALDH1A1HPGDRAB9ATSHR
SCHEMBL31117178 0.89 HTT (0.80) HTTALDH1A1HPGDRAB9ATSHR
SCHEMBL11128807 0.89 HTT (0.80) HTTALDH1A1HPGDRAB9ATSHR
SCHEMBL31117093 0.88 HTT (1.00) HTTALDH1A1HPGDRAB9ATSHR
SCHEMBL10340638 0.88 HTT (1.00) HTTALDH1A1HPGDRAB9ATSHR
SCHEMBL31117075 0.87 HTT (0.77) HTTALDH1A1HPGDRAB9ATSHR
SCHEMBL18987325 0.87 HTT (0.77) HTTALDH1A1HPGDRAB9ATSHR
SCHEMBL31117147 0.87 HTT (0.77) HTTALDH1A1HPGDRAB9ATSHR
SCHEMBL1353689 0.87 HTT (0.77) HTTALDH1A1HPGDRAB9ATSHR
SCHEMBL31117228 0.87 HTT (0.77) HTTALDH1A1HPGDRAB9ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1016398-B The pollen that contains pyrazole derivatives generates composite inhibiting ELLI LILLY & CO (US) 1992-04-29 CN disclosed
EP-0177242-B1 POLLEN FORMATION INHIBITING PYRAZOLES ELI LILLY AND COMPANY (US) 1990-01-03 EP disclosed
US-4775409-A PREVENTING POLLEN FORMATION ELI LILLY AND COMPANY (US) 1988-10-04 US disclosed
US-4666504-A HYBRIDS ELI LILLY AND COMPANY (US) 1987-05-19 US disclosed
CN-85107078-A The pollen that contains pyridine derivate generates composite inhibiting 1987-04-01 CN disclosed
EP-0177242-A2 Pollen formation inhibiting pyrazoles ELI LILLY AND COMPANY (US) 1986-04-09 EP disclosed