SCHEMBL10355381

SCHEMBL10355381

COc1ccc(-c2[nH]cnc2CO)cc1OC

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 4/20 0.49
ALDH1A1 P00352 2/20 0.45
FYN P06241 2/20 0.45
CCNB2 O95067 1/20 0.45
CDK1 P06493 1/20 0.45
CCNB1 P14635 1/20 0.45
GSK3A P49840 1/20 0.45
GSK3B P49841 1/20 0.45
CDK5 Q00535 1/20 0.45
CDK5R1 Q15078 1/20 0.45
CCNB3 Q8WWL7 1/20 0.45
PDGFRB P09619 1/20 0.43
PDGFRA P16234 1/20 0.43
KMT2A Q03164 2/20 0.43
MAPT P10636 2/20 0.43
MEN1 O00255 1/20 0.43
GAA P10253 1/20 0.43
LMNA P02545 1/20 0.43
KDM4E B2RXH2 1/20 0.43
PDE4A P27815 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10355385 0.98 IDO1 (0.48) IDO1ALDH1A1FYNCCNB2CDK1
SCHEMBL10355641 0.83 IDO1 (0.42) IDO1ALDH1A1CCNB2CDK1CCNB1
Hydrochloric Acid SCHEMBL10355404 0.82 IDO1 (0.41) IDO1ALDH1A1CCNB2CDK1CCNB1
SCHEMBL11004015 0.78 DYRK1A (0.47) IDO1FYNCCNB2CDK1CCNB1
Hydrochloric Acid SCHEMBL10355432 0.77 DYRK1A (0.46) IDO1FYNCCNB2CDK1CCNB1
SCHEMBL27915583 0.77 MAPK14 (0.56) IDO1FYNCCNB2CDK1CCNB1
SCHEMBL10355257 0.76 KDM4E (0.39) IDO1MAPTGAAKDM4E
SCHEMBL10355621 0.75 HPGD (0.56) ALDH1A1PDGFRBPDGFRAKMT2AMAPT
SCHEMBL10355357 0.74 IDO1 (0.58) IDO1ALDH1A1FYNCCNB2CDK1
SCHEMBL10355322 0.74 CYP11B1 (0.44) IDO1ALDH1A1KMT2AMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0074130-B1 NEW IMIDAZOLE COMPOUNDS, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM ZAMBON S.p.A. (IT) 1990-09-19 EP disclosed
US-4560696-A Analgesic, antipyretic or anti-inflammatory imidazole compounds ZAMBON S.P.A. (IT) 1985-12-24 US disclosed
EP-0074130-A2 New imidazole compounds, process for the preparation thereof and pharmaceutical compositions containing them ZAMBON S.p.A. (IT) 1983-03-16 EP disclosed