SCHEMBL10356459

SCHEMBL10356459

CCC1COC(c2ccc(C#N)cc2)CO1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 8/20 0.43
CHRM3 P20309 6/20 0.43
CHRM4 P08173 4/20 0.43
CHRM1 P11229 4/20 0.43
CHRM5 P08912 6/20 0.41
CYP2A6 P11509 1/20 0.38
HTR1A P08908 4/20 0.37
ADRA1D P25100 3/20 0.37
ADRA1A P35348 3/20 0.37
TSHR P16473 1/20 0.36
GRIA2 P42262 1/20 0.34
KCNH2 Q12809 1/20 0.34
ADRA1B P35368 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10689277 1.00 CHRM2 (0.43) CHRM2CHRM3CHRM4CHRM1CHRM5
SCHEMBL10689377 0.96 CHRM2 (0.49) CHRM2CHRM3CHRM4CHRM1CHRM5
SCHEMBL10689371 0.96 CHRM2 (0.49) CHRM2CHRM3CHRM4CHRM1CHRM5
SCHEMBL10689386 0.96 CHRM2 (0.49) CHRM2CHRM3CHRM4CHRM1CHRM5
SCHEMBL7508064 0.88 CHRM2 (0.41) CHRM2CHRM3CHRM4CHRM1CHRM5
SCHEMBL8046421 0.88 CHRM2 (0.41) CHRM2CHRM3CHRM4CHRM1CHRM5
SCHEMBL8046424 0.88 CHRM2 (0.41) CHRM2CHRM3CHRM4CHRM1CHRM5
SCHEMBL8449001 0.85 GRM2 (0.43) CHRM2CHRM3CHRM4CHRM1CHRM5
SCHEMBL10687897 0.85 GRM2 (0.43) CHRM2CHRM3CHRM4CHRM1CHRM5
SCHEMBL10688995 0.84 CHRM2 (0.47) CHRM2CHRM3CHRM4CHRM1CHRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0151446-B1 LIQUID CRYSTAL PHASE MERCK PATENT GmbH (DE) 1990-09-19 EP disclosed
US-4755323-A Mixture of liquid crystalline compounds including substituted para-dioxane MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1988-07-05 US disclosed
EP-0151446-A2 Liquid crystal phase MERCK PATENT GmbH (DE) 1985-08-14 EP disclosed