SCHEMBL10360787

SCHEMBL10360787

CC(n1cncn1)C(O)(c1ccc(OC(F)(F)F)cc1)c1ccc(OC(F)(F)F)cc1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 2/20 0.42
POLB P06746 1/20 0.39
CYP19A1 P11511 1/20 0.39
CYP3A4 P08684 1/20 0.38
CCR6 P51684 13/20 0.38
KCNH2 Q12809 7/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
LMNA P02545 1/20 0.36
SCN5A Q14524 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10565684 0.86 CYP19A1 (0.40) HSP90AA1POLBCYP19A1CYP3A4CCR6
SCHEMBL10360756 0.86 HSP90AA1 (0.46) HSP90AA1POLBCYP19A1CYP3A4MEN1
SCHEMBL10565696 0.84 CYP19A1 (0.41) HSP90AA1POLBCYP19A1CYP3A4CCR6
SCHEMBL10360981 0.83 HSP90AA1 (0.46) HSP90AA1CYP19A1CYP3A4KMT2ALMNA
SCHEMBL10361161 0.80 HSP90AA1 (0.46) HSP90AA1POLBCYP19A1CYP3A4MEN1
SCHEMBL10361057 0.80 CYP19A1 (0.51) HSP90AA1POLBCYP19A1CYP3A4MEN1
SCHEMBL10361515 0.80 CYP19A1 (0.46) HSP90AA1POLBCYP19A1CYP3A4MEN1
SCHEMBL10360965 0.80 CCR6 (0.40) CCR6KCNH2SCN5A
SCHEMBL10362206 0.80 HSP90AA1 (0.62) HSP90AA1POLBCYP19A1CYP3A4MEN1
SCHEMBL16731565 0.79 CCR6 (0.39) CCR6KCNH2SCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0158448-B1 AZOLYL PROPANOLS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1990-08-29 EP claimed
EP-0158448-B1 AZOLYL PROPANOLS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1990-08-29 EP disclosed
US-4833159-A FUNGICIDES IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-05-23 US disclosed
US-4829074-A INSECTICIDES IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-05-09 US disclosed
US-4689337-A 1,2,4-TRIAZOLYL AND PYRAZOLYL GROUPS; FUNGICIDES IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1987-08-25 US disclosed
EP-0158448-A2 Azolyl propanols IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1985-10-16 EP disclosed