SCHEMBL10364232

SCHEMBL10364232

COc1cc(I)nc(NC(=O)NS(=O)(=O)c2ccccc2C(=O)O)n1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.51
CDK1 P06493 1/20 0.48
MAPT P10636 3/20 0.44
TP53 P04637 1/20 0.44
GLA P06280 1/20 0.44
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
MMP1 P03956 1/20 0.41
MMP2 P08253 1/20 0.41
MMP9 P14780 1/20 0.41
MMP8 P22894 1/20 0.41
MMP13 P45452 1/20 0.41
KMT2A Q03164 1/20 0.40
KDM4E B2RXH2 1/20 0.40
NPC1 O15118 1/20 0.40
ALDH1A1 P00352 1/20 0.40
CA12 O43570 1/20 0.39
CA9 Q16790 1/20 0.39
TSHR P16473 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10469643 0.92 GAA (0.59) GAACDK1MAPTTP53GLA
SCHEMBL119097 0.88 GAA (0.52) GAACDK1MAPTTP53GLA
SCHEMBL10506007 0.88 TSHR (0.53) GAACDK1MAPTTP53GLA
SCHEMBL29371340 0.88 GAA (0.52) GAACDK1MAPTTP53GLA
SCHEMBL10364239 0.88 CDK1 (0.51) GAACDK1MAPTTP53GLA
SCHEMBL11246536 0.85 CDK1 (0.51) GAACDK1MAPTTP53GLA
SCHEMBL4887087 0.85 GAA (0.49) GAACDK1MAPTTP53GLA
SCHEMBL9200551 0.85 GAA (0.53) GAACDK1MAPTTP53GLA
SCHEMBL10565058 0.85 GAA (0.48) GAACDK1MAPTTP53GLA
SCHEMBL10363991 0.84 GAA (0.50) GAACDK1MAPTTP53GLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0161905-B1 HERBICIDAL HALOPYRIMIDINES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1990-08-01 EP claimed
US-4659361-A PLANT GROWTH REGULATORS E. I. DU PONT DE NEMOURS AND COMPANY (US) 1987-04-21 US claimed
EP-0161905-A2 Herbicidal halopyrimidines E.I. DU PONT DE NEMOURS AND COMPANY (US) 1985-11-21 EP claimed
EP-0161905-B1 HERBICIDAL HALOPYRIMIDINES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1990-08-01 EP disclosed
US-4659361-A PLANT GROWTH REGULATORS E. I. DU PONT DE NEMOURS AND COMPANY (US) 1987-04-21 US disclosed
US-4659361-A PLANT GROWTH REGULATORS E. I. DU PONT DE NEMOURS AND COMPANY (US) 1987-04-21 US disclosed
EP-0161905-A2 Herbicidal halopyrimidines E.I. DU PONT DE NEMOURS AND COMPANY (US) 1985-11-21 EP disclosed