SCHEMBL10367165

SCHEMBL10367165

CC(=O)SCCN1C(=O)c2ccccc2C1=O

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.56
RAB9A P51151 2/20 0.56
SMN1; SMN2 Q16637 2/20 0.56
CASP3 P42574 1/20 0.56
SENP8 Q96LD8 1/20 0.56
SENP7 Q9BQF6 1/20 0.56
SENP6 Q9GZR1 1/20 0.56
KMT2A Q03164 3/20 0.54
MEN1 O00255 2/20 0.54
GAA P10253 1/20 0.54
ALDH1A1 P00352 4/20 0.52
CYP1A2 P05177 2/20 0.52
CYP2C19 P33261 2/20 0.52
HPGD P15428 1/20 0.50
HDAC8 Q9BY41 3/20 0.49
HDAC3 O15379 2/20 0.49
HDAC4 P56524 2/20 0.49
HDAC1 Q13547 2/20 0.49
HDAC7 Q8WUI4 2/20 0.49
HDAC2 Q92769 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9970727 0.90 CYP1A2 (0.58) KMT2AMEN1CYP1A2CYP2C19CYP2D6
SCHEMBL18374069 0.89 CYP1A2 (0.53) KMT2ACYP1A2CYP2C19HDAC8HDAC3
SCHEMBL29387341 0.89 CYP1A2 (0.53) KMT2ACYP1A2CYP2C19HDAC8HDAC3
SCHEMBL30601912 0.87 HDAC8 (0.55) SMN1; SMN2KMT2AMEN1CYP1A2CYP2C19
SCHEMBL29386458 0.87 HDAC8 (0.55) SMN1; SMN2KMT2AMEN1CYP1A2CYP2C19
SCHEMBL25123844 0.87 HDAC8 (0.55) SMN1; SMN2KMT2AMEN1CYP1A2CYP2C19
SCHEMBL29990582 0.87 HDAC8 (0.55) SMN1; SMN2KMT2AMEN1CYP1A2CYP2C19
SCHEMBL29991896 0.87 HDAC8 (0.55) SMN1; SMN2KMT2AMEN1CYP1A2CYP2C19
SCHEMBL25123876 0.87 HDAC8 (0.55) SMN1; SMN2KMT2AMEN1CYP1A2CYP2C19
SCHEMBL18374697 0.87 HDAC8 (0.55) SMN1; SMN2KMT2AMEN1CYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0166697-B1 AROYL SUBSTITUTED DIHYDRO-1,4-THIAZINES CIBA-GEIGY AG (CH) 1990-05-09 EP disclosed
US-4622322-A ANTIRHEUMATIC AGENTS CIBA-GEIGY CORPORATION (US) 1986-11-11 US disclosed
EP-0166697-A2 Aroyl substituted dihydro-1,4-thiazines CIBA-GEIGY AG (CH) 1986-01-02 EP disclosed