SCHEMBL10367274

SCHEMBL10367274

COC(=O)OC1=C(C)NC(C)=C(c2nc(CN(C)CCCc3ccccc3)no2)C1c1cccc([N+](=O)[O-])c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 7/20 0.49
CYP3A4 P08684 7/20 0.49
CYP2C9 P11712 7/20 0.49
CYP2C19 P33261 7/20 0.49
LMNA P02545 6/20 0.49
MAPT P10636 6/20 0.49
CYP2D6 P10635 5/20 0.49
TSHR P16473 4/20 0.49
TDP1 Q9NUW8 3/20 0.49
ADORA3 P0DMS8 2/20 0.49
ADRA1A P35348 2/20 0.49
MTOR P42345 2/20 0.49
RAB9A P51151 2/20 0.49
SLC6A3 Q01959 2/20 0.49
ADRA2A P08913 2/20 0.49
ABCB1 P08183 2/20 0.49
NPC1 O15118 1/20 0.49
ABCC4 O15439 1/20 0.49
ABCB11 O95342 1/20 0.49
PGR P06401 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10370821 0.96 CYP1A2 (0.51) CYP1A2CYP3A4CYP2C9CYP2C19LMNA
SCHEMBL10366475 0.93 CYP1A2 (0.52) CYP1A2CYP3A4CYP2C9CYP2C19LMNA
SCHEMBL10370936 0.92 CYP1A2 (0.54) CYP1A2CYP3A4CYP2C9CYP2C19LMNA
SCHEMBL7317006 0.90 CYP1A2 (0.60) CYP1A2CYP3A4CYP2C9CYP2C19LMNA
SCHEMBL10366346 0.88 CACNA1C (0.50) CYP1A2CYP3A4CYP2C9CYP2C19LMNA
SCHEMBL10366351 0.88 CACNA1C (0.50) CYP1A2CYP3A4CYP2C9CYP2C19LMNA
SCHEMBL10369421 0.88 CYP1A2 (0.47) CYP1A2CYP3A4CYP2C9CYP2C19LMNA
SCHEMBL7271902 0.87 PDE1C (0.48) CYP1A2CYP3A4CYP2C9CYP2C19LMNA
SCHEMBL10375090 0.87 CYP1A2 (0.46) CYP1A2CYP3A4CYP2C9CYP2C19LMNA
SCHEMBL10368720 0.87 CYP1A2 (0.46) CYP1A2CYP3A4CYP2C9CYP2C19LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0177965-B1 NOVEL OXA- AND THIADIAZOLYL DERIVATIVES AND THEIR USE SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1990-03-21 EP claimed