SCHEMBL10368591

SCHEMBL10368591

O=C(O)[C@@H](S)c1ccncc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAPRT Q6XQN6 1/20 0.44
SLC6A2 P23975 2/20 0.43
SLC6A4 P31645 2/20 0.43
SLC6A3 Q01959 2/20 0.43
CYP3A4 P08684 2/20 0.41
CYP2C19 P33261 2/20 0.41
KDM4E B2RXH2 1/20 0.40
HSD17B10 Q99714 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
GRM8 O00222 1/20 0.39
GRM4 Q14833 1/20 0.39
ALDH1A1 P00352 3/20 0.37
MDM2 Q00987 1/20 0.37
AKR1C3 P42330 1/20 0.37
AKR1C2 P52895 1/20 0.37
TAAR1 Q96RJ0 1/20 0.36
PLOD2 O00469 1/20 0.36
PLOD3 O60568 1/20 0.36
CYP1A2 P05177 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1574188 1.00 NAPRT (0.44) NAPRTSLC6A2SLC6A4SLC6A3CYP3A4
Pyridine SCHEMBL28109952 0.85 SRC (0.45) SLC6A2SLC6A4SLC6A3MEN1KMT2A
SCHEMBL997295 0.83 SRC (0.42) CYP2C19KDM4EHSD17B10MEN1KMT2A
SCHEMBL11798536 0.80 CYP3A4 (0.40) NAPRTSLC6A2SLC6A4SLC6A3CYP3A4
Hydrochloric Acid SCHEMBL11299975 0.78 CYP3A4 (0.39) NAPRTSLC6A2SLC6A4SLC6A3CYP3A4
SCHEMBL74366 0.78 SRC (0.56) CYP2C19CYP1A2CYP2D6LMNA
SCHEMBL27264628 0.77 CYP3A4 (0.38) NAPRTSLC6A2SLC6A4SLC6A3CYP3A4
SCHEMBL8062050 0.76 SRC (0.61) NAPRTSLC6A2SLC6A4SLC6A3CYP3A4
Hydrochloric Acid SCHEMBL8340022 0.76 SRC (0.54) CYP1A2CYP2D6LMNA
SCHEMBL7052263 0.75 CYP2D6 (0.43) NAPRTSLC6A2SLC6A4SLC6A3CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0175363-B1 4,5-DIHYDRO-3(2H)-PYRIDAZINONES, PROCESS FOR THEIR PREPARATION AND THEIR USE CASSELLA Aktiengesellschaft (DE) 1990-01-17 EP disclosed
US-4816454-A CARDIOVASCULAR DISORDERS CASSELLA AKTIENGESELLSCHAFT (DE) 1989-03-28 US disclosed
EP-0175363-A2 4,5-Dihydro-3(2H)-pyridazinones, process for their preparation and their use CASSELLA Aktiengesellschaft (DE) 1986-03-26 EP disclosed