SCHEMBL1036867

SCHEMBL1036867

CCOc1ccc(Cc2cc([C@@H]3N[C@H](CO)C(O)[C@H](O)[C@H]3O)ccc2Cl)cc1

nearest known ligand 0.68

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SLC5A2 P31639 19/20 0.68
SLC5A1 P13866 11/20 0.68
ADRA2A P08913 1/20 0.63
SLC5A11 Q8WWX8 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1037836 1.00 SLC5A2 (0.68) SLC5A2SLC5A1ADRA2ASLC5A11
SCHEMBL1036645 1.00 SLC5A2 (0.68) SLC5A2SLC5A1ADRA2ASLC5A11
SCHEMBL2997996 1.00 SLC5A2 (0.68) SLC5A2SLC5A1ADRA2ASLC5A11
SCHEMBL16473307 0.88 SLC5A2 (0.64) SLC5A2SLC5A1ADRA2ASLC5A11
SCHEMBL14188980 0.85 SLC5A2 (0.60) SLC5A2SLC5A1ADRA2ASLC5A11
SCHEMBL1487476 0.81 SLC5A2 (1.00) SLC5A2SLC5A1ADRA2ASLC5A11
SCHEMBL1039664 0.80 SLC5A2 (0.59) SLC5A2SLC5A1ADRA2ASLC5A11
SCHEMBL16457244 0.80 SLC5A2 (0.59) SLC5A2SLC5A1ADRA2ASLC5A11
SCHEMBL16457243 0.80 SLC5A2 (0.59) SLC5A2SLC5A1ADRA2ASLC5A11
SCHEMBL48097 0.79 SLC5A2 (0.67) SLC5A2SLC5A1ADRA2ASLC5A11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2308841-B1 Phlorizin analogs as SGLT2 inhibitors LEXICON PHARMACEUTICALS INC (US) 2014-04-16 EP disclosed
EP-2308841-A2 Phlorizin analogs as SGLT2 inhibitors Lexicon Pharmaceuticals, Inc. (US) 2011-04-13 EP disclosed
EP-2089361-B1 INHIBITORS OF SODIUM GLUCOSE CO-TRANSPORTER 2 AND METHODS OF THEIR USE LEXICON PHARMACEUTICALS INC (US) 2011-01-26 EP disclosed