SCHEMBL10375437

SCHEMBL10375437

CCOC(=O)c1c(C)nc(-c2cccnc2)nc1-c1cc([N+](=O)[O-])ccc1Cl

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
ALDH1A1 P00352 2/20 0.42
MAPK1 P28482 1/20 0.42
DCTPP1 Q9H773 1/20 0.41
KDM4E B2RXH2 3/20 0.41
TP53 P04637 1/20 0.41
RAB9A P51151 1/20 0.41
HSD17B10 Q99714 1/20 0.41
CYP19A1 P11511 3/20 0.41
CYP11B1 P15538 3/20 0.41
CYP11B2 P19099 3/20 0.41
PDE4B Q07343 1/20 0.40
PDE4D Q08499 1/20 0.40
PDE5A O76074 2/20 0.40
CACNB4 O00305 1/20 0.39
CACNA1A O00555 1/20 0.39
CACNA1G O43497 1/20 0.39
CACNG3 O60359 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10375307 0.91 MAPT (0.43) MAPTALDH1A1MAPK1DCTPP1KDM4E
SCHEMBL10375315 0.90 KDM4E (0.52) MAPTALDH1A1MAPK1KDM4ETP53
SCHEMBL10375306 0.88 CACNA1C (0.42) MAPTMEN1KMT2AALDH1A1MAPK1
SCHEMBL10376545 0.86 MAPT (0.49) MAPTMEN1KMT2AALDH1A1MAPK1
SCHEMBL10375516 0.81 KDM4E (0.54) MAPTMEN1KMT2AALDH1A1MAPK1
SCHEMBL10375348 0.81 KMT2A (0.43) MAPTMEN1KMT2AALDH1A1MAPK1
SCHEMBL10375515 0.78 KDM4E (0.50) MAPTALDH1A1MAPK1KDM4ETP53
SCHEMBL10375512 0.77 KDM4E (0.49) MAPTMEN1KMT2AALDH1A1MAPK1
SCHEMBL10375290 0.77 KDM4E (0.49) MAPTALDH1A1MAPK1KDM4ETP53
SCHEMBL10375328 0.76 MAOB (0.44) MAPTMEN1KMT2AALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0169712-B1 NEW PYRIMIDINE DERIVATIVES, PROCESSES FOR PREPARATION THEREOF AND COMPOSITION CONTAINING THE SAME FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1990-12-12 EP disclosed
US-4698340-A TREATMENT OF CEREBROVASCULAR DISEASES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1987-10-06 US disclosed
EP-0169712-A2 New pyrimidine derivatives, processes for preparation thereof and composition containing the same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1986-01-29 EP disclosed