SCHEMBL10376147

SCHEMBL10376147

O=Cc1ccc(OCCCC(=O)N(CCO)C2CCCCC2)cc1[N+](=O)[O-]

nearest known ligand 0.50

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 20/20 0.50
PDE3A Q14432 20/20 0.50
P2RY12 Q9H244 11/20 0.47
PDE2A O00408 7/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10375973 0.97 PDE3B (0.47) PDE3BPDE3AP2RY12PDE2A
SCHEMBL7307471 0.93 PDE3B (0.50) PDE3BPDE3AP2RY12PDE2A
SCHEMBL10376996 0.91 PDE3B (0.49) PDE3BPDE3AP2RY12PDE2A
SCHEMBL10376471 0.91 PDE3B (0.46) PDE3BPDE3AP2RY12PDE2A
SCHEMBL10374470 0.90 PDE3B (0.47) PDE3BPDE3AP2RY12PDE2A
SCHEMBL7317749 0.90 PDE3B (0.46) PDE3BPDE3AP2RY12PDE2A
SCHEMBL7317830 0.90 PDE3B (0.49) PDE3BPDE3AP2RY12PDE2A
SCHEMBL7307541 0.89 PDE3B (0.46) PDE3BPDE3AP2RY12PDE2A
SCHEMBL10374494 0.89 PDE3B (0.47) PDE3BPDE3AP2RY12PDE2A
SCHEMBL10376736 0.87 PDE3B (0.45) PDE3BPDE3AP2RY12PDE2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0116948-B1 (2-OXO-1,2,3,5-TETRAHYDROIMIDAZO-(2,1-B)QUINAZOLINYL)-OXYALKYL-AMIDES SYNTEX (U.S.A.) INC. (US) 1990-01-03 EP disclosed
US-4663320-A ANTITUMOR AGENTS, ANTICOAGULANTS SYNTEX (U.S.A.) INC. (US) 1987-05-05 US disclosed
US-4551459-A Method of treating heart failure using (2-oxo-1,2,3,5-tetrahydroimidazo-[2,1-b]quinazolinyl)oxyalkylamides SYNTEX (U.S.A.) INC. (US) 1985-11-05 US disclosed
US-4490371-A ANTICOAGULANTS, PHOSPHODIESTERASE INHIBITORS SYNTEX (U.S.A.) INC. (US) 1984-12-25 US disclosed
EP-0116948-A2 (2-Oxo-1,2,3,5-tetrahydroimidazo-(2,1-b)quinazolinyl)-oxyalkyl-amides SYNTEX (U.S.A.) INC. (US) 1984-08-29 EP disclosed