SCHEMBL10377774

SCHEMBL10377774

Cc1ccc(-c2nccc3[nH]c(=O)ccc23)cc1

nearest known ligand 0.73

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 18/20 0.73
PDE3A Q14432 18/20 0.73
BCHE P06276 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10377813 0.84 PDE3B (1.00) PDE3BPDE3A
SCHEMBL10378694 0.84 PDE3B (1.00) PDE3BPDE3A
SCHEMBL10378903 0.84 PDE3B (1.00) PDE3BPDE3A
SCHEMBL10378892 0.84 PDE3B (0.73) PDE3BPDE3A
SCHEMBL10379203 0.84 PDE3B (1.00) PDE3BPDE3ABCHE
SCHEMBL10807799 0.84 PDE3B (1.00) PDE3BPDE3A
SCHEMBL2309156 0.84 PDE3B (1.00) PDE3BPDE3A
SCHEMBL10811148 0.84 PDE3B (0.63) PDE3BPDE3A
SCHEMBL10378883 0.84 PDE3B (1.00) PDE3BPDE3ABCHE
SCHEMBL10378576 0.84 PDE3B (0.68) PDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0168037-B1 1-6-NAPHTHYRIDIN-2(1H)-ONES USEFUL AS CARDIOTONICS STERLING DRUG INC. (US) 1990-02-07 EP disclosed
EP-0168037-A2 1-6-Naphthyridin-2(1H)-ones useful as cardiotonics STERLING DRUG INC. (US) 1986-01-15 EP disclosed
US-4560691-A 5-(Phenyl)-1,6-naphthyridin-2(1H)-ones, their cardiotonic use and preparation STERLING DRUG INC. (US) 1985-12-24 US disclosed