SCHEMBL10414720

SCHEMBL10414720

COc1cc2c(cc1OC)C(Oc1ccc(C)cc1)CN(C)CC2

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.55
CYP2D6 P10635 1/20 0.55
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
DPP4 P27487 2/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA9 Q16790 1/20 0.47
CA14 Q9ULX7 1/20 0.47
MAOA P21397 3/20 0.47
MAOB P27338 2/20 0.46
SLC6A4 P31645 1/20 0.46
KCNN2 Q9H2S1 3/20 0.44
KCNN3 Q9UGI6 3/20 0.44
BRD4 O60885 2/20 0.44
KCNN1 Q92952 1/20 0.44
DRD1 P21728 2/20 0.44
DRD5 P21918 2/20 0.44
DRD4 P21917 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9797273 0.92 CYP3A4 (0.57) CYP3A4CYP2D6MAOAMAOBSLC6A4
Hydrochloric Acid SCHEMBL9797260 0.91 CYP3A4 (0.56) CYP3A4CYP2D6MAOAMAOBSLC6A4
Fumaric Acid SCHEMBL9806127 0.90 CYP3A4 (0.49) CYP3A4CYP2D6MEN1KMT2ADPP4
Maleic Acid SCHEMBL9806125 0.90 CYP3A4 (0.49) CYP3A4CYP2D6MEN1KMT2ADPP4
SCHEMBL9797324 0.89 CYP3A4 (0.54) CYP3A4CYP2D6CA1CA2CA9
SCHEMBL9797712 0.89 CYP3A4 (0.54) CYP3A4CYP2D6CA1CA2CA9
SCHEMBL9797470 0.89 CYP3A4 (0.54) CYP3A4CYP2D6MEN1KMT2ACA1
SCHEMBL9797731 0.88 CYP3A4 (0.67) CYP3A4CYP2D6DPP4MAOAMAOB
SCHEMBL9797438 0.85 CYP3A4 (0.51) CYP3A4CYP2D6MEN1KMT2AMAOA
SCHEMBL10416119 0.85 CYP3A4 (0.51) CYP3A4CYP2D6MEN1KMT2ACA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4935418-A Medical compositions of 1-aryloxy-2,3,4,5-tetrahydro-3-benzazepines and use thereof HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1990-06-19 US claimed
US-4794181-A ANTIDEPRESSANTS, ANALGESICS HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1988-12-27 US claimed