SCHEMBL10421985

SCHEMBL10421985

COC(=O)CCCCCNC(=O)C(C)NC(=O)OC(C)(C)C

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
KMT2A Q03164 2/20 0.46
HDAC8 Q9BY41 1/20 0.42
CA1 P00915 2/20 0.42
CA2 P00918 2/20 0.42
CA7 P43166 1/20 0.42
MAOA P21397 1/20 0.42
MAOB P27338 1/20 0.42
MEN1 O00255 1/20 0.41
GAA P10253 1/20 0.41
EPHX2 P34913 4/20 0.41
CTSS P25774 1/20 0.40
CTSK P43235 1/20 0.40
CA12 O43570 1/20 0.39
CA9 Q16790 1/20 0.39
CYP2D6 P10635 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10421986 1.00 CAPN1 (0.47) CAPN1TDP1KMT2AHDAC8CA1
SCHEMBL25449140 1.00 CAPN1 (0.47) CAPN1TDP1KMT2AHDAC8CA1
SCHEMBL12056633 0.94 CAPN1 (0.52) CAPN1TDP1KMT2ACA1CA2
SCHEMBL7346299 0.85 CAPN1 (0.50) CAPN1TDP1KMT2AMAOAMAOB
SCHEMBL24366566 0.83 CAPN1 (0.52) CAPN1KMT2ACA1CA2CA7
SCHEMBL22276594 0.82 TDP1 (0.67) TDP1KMT2ACA1CA2MAOA
SCHEMBL19078966 0.82 TDP1 (0.67) TDP1KMT2ACA1CA2MAOA
SCHEMBL25092096 0.82 TDP1 (0.67) TDP1KMT2ACA1CA2MAOA
SCHEMBL22276612 0.82 TDP1 (0.67) TDP1KMT2ACA1CA2MAOA
SCHEMBL2582992 0.82 TDP1 (0.67) TDP1KMT2ACA1CA2MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4933325-A ANALGESICS, HYPOTENSIVE AGENTS G. D. SEARLE & CO. (US) 1990-06-12 US disclosed
US-4880829-A ANALGESICS, HYPOTENSIVE AGENTS G. D. SEARLE AND COMPANY (US) 1989-11-14 US disclosed
US-4847241-A ANALGESICS G. D. SEARLE & CO. (US) 1989-07-11 US disclosed
US-4822775-A ANALGESICS G. D. SEARLE & CO. (US) 1989-04-18 US disclosed
EP-0215297-A2 Substituted dipeptide amides G.D. Searle & Co. (US) 1987-03-25 EP disclosed