SCHEMBL10422293

SCHEMBL10422293

FCOCOc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNA3 P22001 1/20 0.50
TAAR1 Q96RJ0 1/20 0.44
ALDH1A1 P00352 1/20 0.44
RECQL P46063 1/20 0.44
ALOX15 P16050 1/20 0.43
LTA4H P09960 2/20 0.41
HDAC1 Q13547 2/20 0.40
HDAC2 Q92769 2/20 0.40
HDAC3 O15379 1/20 0.40
HDAC4 P56524 1/20 0.40
HDAC7 Q8WUI4 1/20 0.40
HDAC10 Q969S8 1/20 0.40
HDAC11 Q96DB2 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
HDAC9 Q9UKV0 1/20 0.40
HDAC5 Q9UQL6 1/20 0.40
KCNH2 Q12809 1/20 0.40
DRD2 P14416 1/20 0.40
DRD4 P21917 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5188457 0.84 KCNA3 (0.60) KCNA3TAAR1ALDH1A1RECQLALOX15
SCHEMBL1714596 0.81
SCHEMBL497461 0.81 KCNA3 (0.63) KCNA3TAAR1ALDH1A1RECQLALOX15
Hydrochloric Acid SCHEMBL10555789 0.78 KCNA3 (0.60) KCNA3TAAR1ALDH1A1RECQLALOX15
Hydrochloric Acid SCHEMBL10519295 0.78 KCNA3 (0.60) KCNA3TAAR1ALDH1A1RECQLALOX15
Ammonia Solution, Strong SCHEMBL28919640 0.78 KCNA3 (0.60) KCNA3TAAR1ALDH1A1RECQLALOX15
SCHEMBL6467512 0.78 MAOB (0.53) ALDH1A1LMNA
SCHEMBL10032070 0.76 APP (0.49) LTA4HHDAC6DRD2DRD4DRD3
SCHEMBL4331326 0.76 KCNA3 (0.57) KCNA3TAAR1ALDH1A1RECQLALOX15
SCHEMBL4680217 0.75 KCNA3 (0.50) KCNA3TAAR1ALDH1A1RECQLALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4960767-A ANALGESICS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1990-10-02 US disclosed
EP-0353631-A2 Isoxazolobenzoxazepines, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1990-02-07 EP disclosed
US-4873234-A ANALGESICS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1989-10-10 US disclosed