SCHEMBL10476136

SCHEMBL10476136

Fc1ccc(CSc2c(Cl)ccc3c2CCNCC3)cc1F

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 9/20 0.49
HTR2B P41595 9/20 0.49
HTR2A P28223 7/20 0.49
CYP2D6 P10635 2/20 0.38
MLNR O43193 2/20 0.38
PNMT P11086 2/20 0.38
ADRA2A P08913 1/20 0.38
ADRA2B P18089 1/20 0.38
ADRA2C P18825 1/20 0.38
CYP1A2 P05177 1/20 0.37
HIF1A Q16665 1/20 0.37
DAO P14920 2/20 0.36
METAP2 P50579 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
MAOB P27338 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL10476310 0.91 HTR2C (0.41) HTR2CHTR2BHTR2ACYP2D6MLNR
SCHEMBL10476250 0.89 HTR2A (0.47) HTR2CHTR2BHTR2ACYP2D6PNMT
SCHEMBL10228938 0.87 HTR2A (0.49) HTR2CHTR2BHTR2ACYP2D6PNMT
SCHEMBL10228933 0.86 HTR2C (0.48) HTR2CHTR2BHTR2ACYP2D6MLNR
SCHEMBL10476234 0.86 HTR2C (0.50) HTR2CHTR2BHTR2AMLNRPNMT
SCHEMBL10229002 0.86 HTR2C (0.40) HTR2CHTR2BHTR2ACYP2D6PNMT
SCHEMBL10476286 0.85 HTR2C (0.47) HTR2CHTR2BHTR2ACYP2D6MLNR
Hydrochloric Acid SCHEMBL508526 0.85 HTR2C (0.39) HTR2CHTR2BHTR2ACYP2D6PNMT
SCHEMBL10229012 0.85 HTR2A (0.39) HTR2CHTR2BHTR2ACYP2D6PNMT
SCHEMBL10476290 0.84 HTR2C (0.43) HTR2CHTR2BHTR2APNMTADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8580780-B2 6 substituted 2, 3,4,5 tetrahydro-1H-benzo[d]azepines as 5-HT2C receptor agonist ELI LILLY AND COMPANY (US) 2013-11-12 US claimed
EP-2479168-A1 6-Substituted 2,3,4,5-Tetrahydro-1H-Benzo [d]Azepines as 5-HT2C Receptor Agonists ELI LILLY AND COMPANY (US) 2012-07-25 EP claimed