SCHEMBL10476293

SCHEMBL10476293

CCC(=O)c1ccc(CSc2c(Cl)ccc3c2CCNCC3)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 7/20 0.41
HTR2C P28335 7/20 0.41
HTR2B P41595 7/20 0.41
PNMT P11086 2/20 0.35
ADRA2A P08913 1/20 0.35
ADRA2B P18089 1/20 0.35
ADRA2C P18825 1/20 0.35
OPRM1 P35372 2/20 0.34
OPRD1 P41143 2/20 0.34
OPRK1 P41145 2/20 0.34
LMNA P02545 2/20 0.33
HPGD P15428 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
MAPT P10636 1/20 0.33
RAB9A P51151 1/20 0.32
MAPK1 P28482 1/20 0.31
STAT3 P40763 1/20 0.31
ACHE P22303 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10476307 0.99 HTR2A (0.40) HTR2AHTR2CHTR2BPNMTADRA2A
SCHEMBL10476265 0.91 HTR2A (0.39) HTR2AHTR2CHTR2BPNMTADRA2A
Hydrochloric Acid SCHEMBL10476273 0.90 HTR2A (0.39) HTR2AHTR2CHTR2BPNMTADRA2A
SCHEMBL10230342 0.89 HTR2A (0.43) HTR2AHTR2CHTR2BPNMTADRA2A
SCHEMBL10229062 0.88 HTR2A (0.39) HTR2AHTR2CHTR2BPNMTADRA2A
SCHEMBL10476251 0.88 HTR2A (0.39) HTR2AHTR2CHTR2BPNMTADRA2A
Hydrochloric Acid SCHEMBL506926 0.88 HTR2A (0.42) HTR2AHTR2CHTR2BPNMTADRA2A
Hydrochloric Acid SCHEMBL507277 0.87 HTR2A (0.38) HTR2AHTR2CHTR2BPNMTADRA2A
Hydrochloric Acid SCHEMBL10476283 0.87 HTR2A (0.38) HTR2AHTR2CHTR2BPNMTADRA2A
SCHEMBL10476197 0.86 HTR2A (0.40) HTR2AHTR2CHTR2BPNMTADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8580780-B2 6 substituted 2, 3,4,5 tetrahydro-1H-benzo[d]azepines as 5-HT2C receptor agonist ELI LILLY AND COMPANY (US) 2013-11-12 US claimed
EP-2479168-A1 6-Substituted 2,3,4,5-Tetrahydro-1H-Benzo [d]Azepines as 5-HT2C Receptor Agonists ELI LILLY AND COMPANY (US) 2012-07-25 EP claimed