SCHEMBL10488356

SCHEMBL10488356

COCC(C)(CO)NCc1c2ccccc2cc2ccccc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.39
NPBWR1 P48145 1/20 0.39
MCHR1 Q99705 1/20 0.39
CD274 Q9NZQ7 1/20 0.37
HTR2A P28223 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
SLC2A1 P11166 1/20 0.36
ALDH1A1 P00352 3/20 0.36
CYP1A2 P05177 3/20 0.36
HIF1A Q16665 2/20 0.36
ALOX12 P18054 1/20 0.36
PHLPP2 Q6ZVD8 1/20 0.36
HSD17B10 Q99714 1/20 0.36
MEN1 O00255 1/20 0.35
HPGD P15428 2/20 0.34
ABCB1 P08183 1/20 0.33
EDNRA P25101 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10488185 0.99 KMT2A (0.41) KMT2ANPBWR1MCHR1CD274HTR2A
SCHEMBL10488406 0.88 HTR2A (0.43) KMT2ANPBWR1MCHR1CD274HTR2A
Hydrochloric Acid SCHEMBL10488372 0.87 KMT2A (0.43) KMT2ANPBWR1MCHR1CD274HTR2A
SCHEMBL10547740 0.84 SLC2A1 (0.47) KMT2ANPBWR1MCHR1CD274SLC2A1
SCHEMBL10488510 0.83 HTR2A (0.39) KMT2ANPBWR1MCHR1CD274HTR2A
SCHEMBL10348808 0.83 KMT2A (0.40) KMT2ANPBWR1MCHR1CD274HTR2A
Hydrochloric Acid SCHEMBL10546808 0.83 SLC2A1 (0.46) KMT2ANPBWR1MCHR1CD274SLC2A1
SCHEMBL9466082 0.80 CD274 (0.41) KMT2ANPBWR1MCHR1CD274SLC2A1
Hydrochloric Acid SCHEMBL9465698 0.80 KMT2A (0.42) KMT2ANPBWR1MCHR1CD274SLC2A1
SCHEMBL10348691 0.80 SLC2A1 (0.39) KMT2ANPBWR1MCHR1CD274HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0125702-B1 POLYCYCLIC AROMATIC COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1987-08-12 EP claimed
EP-0125702-A2 Polycyclic aromatic compounds THE WELLCOME FOUNDATION LIMITED (GB) 1984-11-21 EP claimed
US-4803221-A Anthracene derivatives BURROUGHS WELLCOME CO. (US) 1989-02-07 US disclosed
US-4719049-A ANTITUMOR BURROUGHS WELLCOME CO. (US) 1988-01-12 US disclosed
EP-0125702-B1 POLYCYCLIC AROMATIC COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1987-08-12 EP disclosed
EP-0125702-A2 Polycyclic aromatic compounds THE WELLCOME FOUNDATION LIMITED (GB) 1984-11-21 EP disclosed