SCHEMBL10488449

SCHEMBL10488449

N#Cc1cccc2c(C=O)c3ccccc3cc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 4/20 0.50
CA2 P00918 4/20 0.50
HTT P42858 2/20 0.44
ERN1 O75460 2/20 0.42
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
CLK1 P49759 1/20 0.39
DYRK1A Q13627 1/20 0.39
MCL1 Q07820 1/20 0.38
ALDH1A1 P00352 3/20 0.38
KDM4E B2RXH2 2/20 0.38
PADI4 Q9UM07 1/20 0.38
MAOA P21397 1/20 0.37
NCOA3 Q9Y6Q9 1/20 0.37
MAPT P10636 3/20 0.36
KDM2B Q8NHM5 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10348702 0.80 ERN1 (0.55) ERN1MEN1KMT2AALDH1A1KDM4E
Acetonitrile SCHEMBL29204821 0.79 ERN1 (0.47) CA1CA2ERN1MEN1KMT2A
SCHEMBL11309875 0.79 ERN1 (0.49) CA1CA2HTTERN1MEN1
SCHEMBL59702 0.78 CA1 (0.69) CA1CA2HTTCLK1DYRK1A
SCHEMBL342278 0.78 ERN1 (0.57) ERN1MEN1KMT2AALDH1A1KDM4E
SCHEMBL29388184 0.78 ERN1 (0.57) ERN1MEN1KMT2AALDH1A1KDM4E
SCHEMBL18322219 0.78 HTT (0.53) CA1CA2HTTCLK1DYRK1A
SCHEMBL1428240 0.77 ERN1 (0.55) CA1CA2HTTERN1MCL1
SCHEMBL1573749 0.77 CA1 (0.50) CA1CA2HTTMEN1KMT2A
SCHEMBL985197 0.77 ERN1 (0.46) ERN1MEN1KMT2AALDH1A1PADI4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4803226-A ANTITUMOR AGENTS BURROUGHS WELLCOME CO. (US) 1989-02-07 US disclosed
US-4803221-A Anthracene derivatives BURROUGHS WELLCOME CO. (US) 1989-02-07 US disclosed
US-4719047-A ANTITUMOR BURROUGHS WELLCOME CO. (US) 1988-01-12 US disclosed
US-4719049-A ANTITUMOR BURROUGHS WELLCOME CO. (US) 1988-01-12 US disclosed