SCHEMBL10517855

SCHEMBL10517855

CCN(CC)CCCCC1CCCN(CCCC(=O)N2c3ccccc3C(=O)Nc3cccnc32)C1

nearest known ligand 0.73

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 6/20 0.73
CHRM4 P08173 3/20 0.73
CHRM1 P11229 3/20 0.73
CHRM3 P20309 3/20 0.73
CHRM5 P08912 1/20 0.73
ALOX15 P16050 1/20 0.73
DRD1 P21728 1/20 0.73
DRD5 P21918 1/20 0.73
TMEM97 Q5BJF2 1/20 0.73
CYP1A2 P05177 1/20 0.56
CYP3A4 P08684 1/20 0.56
MAPK1 P28482 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10518059 0.98 CHRM2 (0.69) CHRM2CHRM4CHRM1CHRM3CHRM5
SCHEMBL10518480 0.94 CHRM2 (0.64) CHRM2CHRM4CHRM1CHRM3CHRM5
SCHEMBL10515620 0.94 CHRM2 (0.65) CHRM2CHRM4CHRM1CHRM3CHRM5
SCHEMBL10515020 0.90
SCHEMBL10516489 0.90 CHRM2 (0.70) CHRM2CHRM4CHRM1CHRM3CHRM5
SCHEMBL10516759 0.89 CHRM2 (0.80) CHRM2CHRM4CHRM1CHRM3CHRM5
SCHEMBL10569796 0.89 CHRM2 (0.67) CHRM2CHRM4CHRM1CHRM3CHRM5
Hydrochloric Acid SCHEMBL9824570 0.88 CHRM2 (0.66) CHRM2CHRM4CHRM1CHRM3CHRM5
SCHEMBL10515636 0.88
Hydrochloric Acid SCHEMBL9676447 0.85 CHRM2 (0.70) CHRM2CHRM4CHRM1CHRM3CHRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0345629-A2 Condensed diazepinones, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1989-12-13 EP disclosed