SCHEMBL10522671

SCHEMBL10522671

C[C@H](CCC(=O)O)[C@H]1CC[C@H]2[C@@H]3[C@H](O)C[C@@H]4C[C@H](OC(=O)CCCCCN(CCCl)CCCl)CC[C@]4(C)[C@H]3C[C@H](O)[C@]12C

nearest known ligand 0.63

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 6/20 0.63
CYP3A4 P08684 3/20 0.63
NR1H4 Q96RI1 3/20 0.63
PDE3A Q14432 1/20 0.63
LMNA P02545 2/20 0.59
KMT2A Q03164 3/20 0.56
MEN1 O00255 2/20 0.56
SLCO1B3 Q9NPD5 1/20 0.56
SLCO1B1 Q9Y6L6 1/20 0.56
USP2 O75604 1/20 0.56
ABCB11 O95342 1/20 0.54
ALDH1A1 P00352 1/20 0.53
TDP1 Q9NUW8 1/20 0.53
SLC10A1 Q14973 1/20 0.51
CYP8B1 Q9UNU6 1/20 0.50
CYP2C19 P33261 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10691725 0.91 GPBAR1 (0.61) GPBAR1CYP3A4NR1H4LMNAKMT2A
SCHEMBL10520272 0.91 GPBAR1 (0.67) GPBAR1CYP3A4NR1H4PDE3ALMNA
SCHEMBL10525788 0.88 GPBAR1 (0.63) GPBAR1CYP3A4NR1H4LMNAKMT2A
SCHEMBL10613228 0.88 GPBAR1 (0.71) GPBAR1CYP3A4NR1H4PDE3ALMNA
SCHEMBL10522119 0.86 CA1 (0.58) GPBAR1CYP3A4NR1H4PDE3AKMT2A
SCHEMBL10520513 0.86 GPBAR1 (0.73) GPBAR1CYP3A4NR1H4PDE3ALMNA
SCHEMBL10521010 0.86 GPBAR1 (0.64) GPBAR1NR1H4PDE3ALMNAKMT2A
SCHEMBL742923 0.85 GPBAR1 (0.65) GPBAR1CYP3A4NR1H4PDE3ALMNA
SCHEMBL23231225 0.85 GPBAR1 (0.83) GPBAR1CYP3A4NR1H4PDE3ALMNA
SCHEMBL21114412 0.85 GPBAR1 (0.83) GPBAR1CYP3A4NR1H4PDE3ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4810422-A CARCINOSTATS OF LOW TOXICITY WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1989-03-07 US disclosed
EP-0259185-A1 Bile acid derivatives, their salts and production thereof WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1988-03-09 EP disclosed