SCHEMBL10530409

SCHEMBL10530409

CC1(C)OC(=O)Nc2cc3nc(-c4cccs4)[nH]c3cc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.47
ALDH1A1 P00352 5/20 0.47
HPGD P15428 4/20 0.47
RAB9A P51151 4/20 0.47
SMN1; SMN2 Q16637 4/20 0.47
TP53 P04637 4/20 0.47
NPC1 O15118 3/20 0.47
MAPT P10636 3/20 0.47
GAA P10253 2/20 0.47
GLA P06280 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
HSD17B10 Q99714 4/20 0.46
KLK7 P49862 1/20 0.46
PDE4A P27815 1/20 0.45
PDE4B Q07343 1/20 0.45
PDE4C Q08493 1/20 0.45
PDE4D Q08499 1/20 0.45
PDE3B Q13370 1/20 0.45
PDE3A Q14432 1/20 0.45
HDAC3 O15379 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10532573 0.81 PDE4A (0.54) KDM4EALDH1A1HPGDRAB9ASMN1; SMN2
SCHEMBL10532459 0.81 PDE4A (0.69) KDM4EALDH1A1HPGDRAB9ANPC1
SCHEMBL10645974 0.80 PDE4A (0.50) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9380784 0.80 KDM4E (0.47) KDM4EALDH1A1HPGDRAB9ASMN1; SMN2
SCHEMBL10530446 0.79 CHEK1 (0.49) KDM4EALDH1A1HPGDRAB9ASMN1; SMN2
SCHEMBL10566333 0.78 PDE4A (0.59) KDM4EALDH1A1HPGDRAB9ASMN1; SMN2
SCHEMBL10534267 0.78 CBFB (0.54) KDM4EALDH1A1HPGDRAB9ASMN1; SMN2
SCHEMBL10532013 0.77 PDE4A (0.52) ALDH1A1HPGDSMN1; SMN2HSD17B10PDE4A
SCHEMBL10532194 0.77 AURKA (0.45) KDM4EALDH1A1HPGDRAB9ASMN1; SMN2
SCHEMBL10534246 0.76 PDE4A (0.48) PDE4APDE4BPDE4CPDE4DPDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4831027-A USEFUL IN TREATMENT OF CARDIOVASCULAR DISORDERS DR. KARL THOMAE GMBH (DE) 1989-05-16 US disclosed