SCHEMBL10552148

SCHEMBL10552148

FC(F)(F)c1cccc(C2=CCNc3ccnn32)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 2/20 0.44
NOTUM Q6P988 2/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
IDO1 P14902 1/20 0.40
SCN2A Q99250 2/20 0.39
PTAFR P25105 1/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
HRH1 P35367 1/20 0.39
HRH4 Q9H3N8 1/20 0.39
CNR2 P34972 1/20 0.38
EPHX2 P34913 1/20 0.38
NR3C1 P04150 1/20 0.38
PGR P06401 1/20 0.38
PARP10 Q53GL7 1/20 0.37
PARP11 Q9NR21 1/20 0.37
HPGD P15428 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
NPY5R Q15761 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5438561 0.82 MAPT (0.52) RAB9A
SCHEMBL9468851 0.79 HPGD (0.41) HTR2CKDM4EALDH1A1IDO1SCN2A
SCHEMBL10461071 0.79 RPS6KB1 (0.40) HTR2CKDM4EALDH1A1IDO1SCN2A
SCHEMBL9468466 0.76 KDM4E (0.50) HTR2CKDM4EALDH1A1IDO1SCN2A
SCHEMBL9870769 0.75 KDM4E (0.43) KDM4EALDH1A1NPC1RAB9AHPGD
SCHEMBL8337425 0.74 KDM4E (0.52) KDM4EALDH1A1NPC1RAB9ANR3C1
SCHEMBL10554628 0.72 CNR2 (0.44) KDM4EALDH1A1NPC1RAB9ACNR2
SCHEMBL10557157 0.72 POLB (0.44) HTR2CKDM4EALDH1A1HPGDSMN1; SMN2
SCHEMBL10557976 0.71 CSNK1E (0.42) KDM4EALDH1A1SMN1; SMN2
SCHEMBL5442258 0.70 DDR2 (0.53)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4847256-A HYPOTENSIVE AGENTS AMERICAN CYANAMID COMPANY (US) 1989-07-11 US disclosed
EP-0264773-A1 4,5-dihydro and 4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidines AMERICAN CYANAMID COMPANY (US) 1988-04-27 EP disclosed