SCHEMBL10575201

SCHEMBL10575201

CCCC1CC2(NC(=O)NC2=O)c2cc(Cl)ccc2O1

nearest known ligand 0.55

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 10/20 0.47
AKR1B10 O60218 2/20 0.46
AKR1A1 P14550 2/20 0.46
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10573588 0.93 AKR1B1 (0.45) AKR1B1AKR1B10AKR1A1MAPT
SCHEMBL10579227 0.91 AKR1B1 (0.43) AKR1B1AKR1B10AKR1A1
SCHEMBL10576212 0.91 AKR1B1 (0.48) AKR1B1AKR1B10AKR1A1MAPT
SCHEMBL10571505 0.86 AKR1B1 (0.62) AKR1B1AKR1B10AKR1A1MAPT
SCHEMBL10578197 0.85 AKR1B1 (0.46) AKR1B1AKR1B10AKR1A1MAPT
SCHEMBL10373488 0.82 AKR1B1 (0.63) AKR1B1AKR1B10AKR1A1
SCHEMBL10576515 0.79 AKR1B1 (0.59) AKR1B1AKR1B10AKR1A1MAPT
SCHEMBL10575580 0.79 AKR1B1 (0.48) AKR1B1AKR1B10AKR1A1MAPT
SCHEMBL10574757 0.77 AKR1B1 (0.65) AKR1B1AKR1B10AKR1A1MAPT
SCHEMBL10574425 0.76 AKR1B1 (0.47) AKR1B1AKR1B10AKR1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4874869-A TREATMENT OF DIABETIC COMPLICATIONS, CATARACTS EISAI CO., LTD. (JP) 1989-10-17 US disclosed
US-4780472-A Hydantoin derivatives for treating complications of diabetes EISAI CO., LTD. (JP) 1988-10-25 US disclosed
US-4540704-A Treating complications of diabetes mellitus with hydantoin derivatives EISAI CO., LTD. (JP) 1985-09-10 US disclosed