SCHEMBL10580909

SCHEMBL10580909

N#Cc1ccc(C=Cc2ccccc2)c(Cn2cncn2)c1

nearest known ligand 0.61

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 19/20 0.61
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10580900 1.00 CYP19A1 (0.61) CYP19A1ALDH1A1HPGD
SCHEMBL10584812 0.93 CYP19A1 (0.56) CYP19A1
SCHEMBL10584822 0.93 CYP19A1 (0.56) CYP19A1
SCHEMBL10583517 0.79 CYP19A1 (0.52) CYP19A1
SCHEMBL10583527 0.79 CYP19A1 (0.52) CYP19A1
SCHEMBL4787857 0.78 CYP19A1 (0.81) CYP19A1
SCHEMBL10172832 0.76 CYP19A1 (1.00) CYP19A1
SCHEMBL10583639 0.71 CYP11B1 (0.56) CYP19A1
SCHEMBL10583642 0.71 CYP11B1 (0.56) CYP19A1
SCHEMBL7061036 0.70 CYP11B1 (0.57) CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0299683-A2 Heterocyclic olefinic compounds and their use as aromatase inhibitors IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-01-18 EP claimed