SCHEMBL10583239

SCHEMBL10583239

COc1ccc(CC(=O)CC(N)=O)cc1

nearest known ligand 0.73

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.61
ALDH1A1 P00352 2/20 0.55
CYP3A4 P08684 1/20 0.55
CYP2C19 P33261 1/20 0.55
F2RL1 P55085 1/20 0.54
SMN1; SMN2 Q16637 2/20 0.51
KDM4E B2RXH2 1/20 0.51
POLB P06746 1/20 0.51
PKM P14618 2/20 0.50
NPC1 O15118 1/20 0.50
MAPK8 P45983 1/20 0.50
CTBP2 P56545 1/20 0.50
LMNA P02545 1/20 0.50
TDP1 Q9NUW8 1/20 0.49
EPHX2 P34913 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31116682 0.85 HTT (0.63) HTTALDH1A1CYP3A4CYP2C19SMN1; SMN2
SCHEMBL1067193 0.85 HTT (0.63) HTTALDH1A1CYP3A4CYP2C19SMN1; SMN2
SCHEMBL3628705 0.85 HTT (0.68) HTTALDH1A1CYP3A4CYP2C19F2RL1
SCHEMBL5431221 0.84 HTT (0.62) HTTALDH1A1CYP3A4CYP2C19F2RL1
SCHEMBL10577487 0.84 HTT (0.62) HTTALDH1A1F2RL1SMN1; SMN2KDM4E
SCHEMBL3280882 0.84 HTT (0.62) HTTALDH1A1F2RL1SMN1; SMN2KDM4E
SCHEMBL6290388 0.81 HTT (0.59) HTTALDH1A1CYP3A4CYP2C19F2RL1
SCHEMBL3175977 0.79 HTT (0.61) HTTALDH1A1CYP3A4CYP2C19F2RL1
SCHEMBL7153605 0.79 HTT (0.61) HTTALDH1A1CYP3A4CYP2C19F2RL1
SCHEMBL14274253 0.78 HTT (0.65) HTTALDH1A1CYP3A4CYP2C19SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0312960-A2 Method for reducing reperfusion injury with imidazol-2-thione-carboxamides MERRELL DOW PHARMACEUTICALS INC. (US) 1989-04-26 EP disclosed