SCHEMBL10632529

SCHEMBL10632529

Oc1cccc(C(O)CN2CCNCC2c2ccccc2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 2/20 0.43
SLC6A3 Q01959 2/20 0.43
SLC6A2 P23975 1/20 0.43
SLC6A4 P31645 1/20 0.43
OPRM1 P35372 2/20 0.40
OPRD1 P41143 2/20 0.40
SLC18A3 Q16572 1/20 0.38
SIGMAR1 Q99720 1/20 0.38
DRD2 P14416 2/20 0.38
DRD3 P35462 2/20 0.37
HIF1A Q16665 2/20 0.37
ADRB2 P07550 1/20 0.37
ADRB1 P08588 1/20 0.37
HTR1A P08908 1/20 0.37
ADRA2A P08913 1/20 0.37
ADRB3 P13945 1/20 0.37
TSHR P16473 1/20 0.37
ADRA2B P18089 1/20 0.37
ADRA2C P18825 1/20 0.37
NFKB1 P19838 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10627836 0.93 SLC6A2 (0.43) CHRNA7SLC6A3SLC6A2SLC6A4OPRM1
SCHEMBL350930 0.89 SLC18A3 (0.44) OPRM1OPRD1SLC18A3SIGMAR1GRIN2B
SCHEMBL10632281 0.87 SLC6A2 (0.42) SLC6A3SLC6A2SLC6A4SLC18A3SIGMAR1
SCHEMBL10630089 0.82 SLC18A3 (0.43) SLC6A3SLC6A2SLC6A4SLC18A3SIGMAR1
SCHEMBL10626688 0.82 GRIN2B (0.35) OPRM1OPRD1SLC18A3SIGMAR1HTR7
SCHEMBL10632309 0.81 SLC18A3 (0.43) SLC18A3SIGMAR1TSHRADRA1AADRA1B
Hydrochloric Acid SCHEMBL10632236 0.81 SLC18A3 (0.43) SLC6A3SLC6A2SLC6A4SLC18A3SIGMAR1
SCHEMBL10627896 0.81 KDM4E (0.39) SLC6A3SLC6A2SLC6A4OPRM1SLC18A3
SCHEMBL10627969 0.80 GRIN2B (0.50) SLC6A2SLC6A4OPRM1OPRD1DRD2
SCHEMBL10627784 0.78 SLC6A2 (0.41) SLC6A2SLC6A4SLC18A3GRIN2BKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4772705-A Processes for the preparation of trans 1,3,4,6,7,11b-hexahydro-7-aryl-2H-pyrazinol[2,1-a]isoquinolines PENNWALT CORPORATION (US) 1988-09-20 US disclosed