SCHEMBL10638592

SCHEMBL10638592

CCOC(=O)c1ccc(C(=O)c2[nH]c(=O)[nH]c2C)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 6/20 0.60
PDE4B Q07343 6/20 0.60
PDE4C Q08493 6/20 0.60
PDE4D Q08499 6/20 0.60
HPGD P15428 5/20 0.60
CYP1A2 P05177 2/20 0.60
CYP3A4 P08684 2/20 0.60
HSD17B10 Q99714 2/20 0.60
PDE3B Q13370 2/20 0.60
PDE3A Q14432 2/20 0.60
NPSR1 Q6W5P4 2/20 0.60
CYP2C9 P11712 1/20 0.60
ALOX15 P16050 1/20 0.60
TSHR P16473 1/20 0.60
NFKB1 P19838 1/20 0.60
BLM P54132 1/20 0.60
PMP22 Q01453 1/20 0.60
ATM Q13315 1/20 0.60
ALDH1A1 P00352 4/20 0.52
RAB9A P51151 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10632401 0.85 PDE3B (0.63) PDE4APDE4BPDE4CPDE4DHPGD
SCHEMBL5457259 0.82 PDE4A (0.53) PDE4APDE4BPDE4CPDE4DHPGD
SCHEMBL3017686 0.80 CYP1A2 (0.58) PDE4DHPGDCYP1A2HSD17B10CYP2C9
SCHEMBL10635511 0.79 PDE4A (0.69) PDE4APDE4BPDE4CPDE4DHPGD
SCHEMBL5457930 0.79 PDE4A (0.69) PDE4APDE4BPDE4CPDE4DHPGD
SCHEMBL8207668 0.78 PDE4A (0.63) PDE4APDE4BPDE4CPDE4DHPGD
SCHEMBL6788089 0.78 CA1 (0.73) HPGDCYP1A2CYP3A4NPSR1TSHR
SCHEMBL11181578 0.78 PDE4A (0.67) PDE4APDE4BPDE4CPDE4DHPGD
SCHEMBL10924200 0.78 PDE4A (0.67) PDE4APDE4BPDE4CPDE4DHPGD
SCHEMBL7339645 0.78 PDE4A (0.67) PDE4APDE4BPDE4CPDE4DHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0118790-B1 NOVEL AROYLIMIDAZOLONES MERRELL DOW PHARMACEUTICALS INC. (US) 1988-07-06 EP disclosed
US-4552880-A Aroylimidazolones MERRELL DOW PHARMACEUTICALS INC. (US) 1985-11-12 US disclosed
EP-0118790-A1 Novel aroylimidazolones MERRELL DOW PHARMACEUTICALS INC. (US) 1984-09-19 EP disclosed