SCHEMBL10649489

SCHEMBL10649489

CN(Cc1ccccc1)C(=O)CCC(=O)c1cccc2c1CN(CC(=O)OOc1ccccc1Cl)C(N)=N2

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
KMT2A Q03164 3/20 0.35
MEN1 O00255 1/20 0.35
AOC3 Q16853 4/20 0.34
L3MBTL1 Q9Y468 1/20 0.33
HPGD P15428 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HSP90AA1 P07900 1/20 0.33
PDE4A P27815 2/20 0.32
PDE4B Q07343 2/20 0.32
PDE4C Q08493 2/20 0.32
PDE4D Q08499 2/20 0.32
CXCR3 P49682 1/20 0.32
PDE3B Q13370 1/20 0.32
PDE3A Q14432 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7313605 0.88 PDE4A (0.40) KMT2AMEN1PDE4APDE4BPDE4C
SCHEMBL10649438 0.85 PDE4A (0.32) PDE4APDE4BPDE4CPDE4D
SCHEMBL10649789 0.85 NPC1 (0.38) NPC1RAB9AKMT2AMEN1L3MBTL1
SCHEMBL10649609 0.80 NPC1 (0.38) NPC1RAB9AKMT2AMEN1L3MBTL1
SCHEMBL10648123 0.78 KMT2A (0.39) NPC1RAB9AKMT2AMEN1HPGD
SCHEMBL7308357 0.74 PDE3B (0.36) NPC1RAB9AKMT2AMEN1HPGD
SCHEMBL7321069 0.74 PDE4A (0.43) KMT2AMEN1L3MBTL1PDE4APDE4B
SCHEMBL7311174 0.73 PDE4A (0.40) NPC1PDE4APDE4BPDE4CPDE4D
SCHEMBL10665307 0.72 PDE4A (0.40) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL7306426 0.71 PDE4A (0.40) KMT2AMEN1PDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0254327-A2 N-N-disubstituted-omega-(2-amino-3-(carbonylmethyl)-3,4-dihydroquinazolinyl) oxyalkylamides and related compounds SYNTEX (U.S.A.) INC. (US) 1988-01-27 EP disclosed