SCHEMBL10654776

SCHEMBL10654776

CCOc1noc2c1CNCC2

nearest known ligand 0.97

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 15/20 0.97
CHRM5 P08912 9/20 0.83
CHRM1 P11229 9/20 0.83
CHRM2 P08172 8/20 0.83
CHRM4 P08173 8/20 0.83
HTR2C P28335 2/20 0.79
HTR2A P28223 1/20 0.79

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10652956 0.98 CHRM3 (1.00) CHRM3CHRM5CHRM1CHRM2CHRM4
SCHEMBL10459676 0.91 CHRM3 (1.00) CHRM3CHRM5CHRM1CHRM2CHRM4
Hydrochloric Acid SCHEMBL10460271 0.89 CHRM3 (0.97) CHRM3CHRM5CHRM1CHRM2CHRM4
SCHEMBL10844384 0.88 CHRM3 (0.97) CHRM3CHRM5CHRM1CHRM2CHRM4
Hydrochloric Acid SCHEMBL10436741 0.87 HTR2C (0.97) CHRM3CHRM5CHRM1CHRM2CHRM4
Hydrochloric Acid SCHEMBL10652707 0.86 CHRM3 (1.00) CHRM3CHRM5CHRM1CHRM2CHRM4
SCHEMBL10654976 0.85 CHRM3 (0.82) CHRM3CHRM5CHRM1CHRM2CHRM4
Hydrochloric Acid SCHEMBL10651499 0.84 CHRM3 (0.84) CHRM3CHRM5CHRM1CHRM2CHRM4
SCHEMBL10655531 0.83 CHRM3 (0.97) CHRM3CHRM5CHRM1CHRM2CHRM4
SCHEMBL10651354 0.81 CHRM3 (0.97) CHRM3CHRM5CHRM1CHRM2CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0126654-B1 TETRAHYDROISOXAZOLO(4,5-C)PYRIDINE DERIVATIVES AND PREPARATION THEREOF H. LUNDBECK A/S (DK) 1988-05-04 EP claimed
US-4608378-A Tetrahydroisoxazolo[4,5-c]pyridine derivatives useful in the treatment of malfunctions of the acetylcholine or muscarinic systems H. LUNDBECK A/S (DK) 1986-08-26 US claimed
EP-0126654-A1 Tetrahydroisoxazolo(4,5-c)pyridine derivatives and preparation thereof H. LUNDBECK A/S (DK) 1984-11-28 EP claimed
EP-0126654-B1 TETRAHYDROISOXAZOLO(4,5-C)PYRIDINE DERIVATIVES AND PREPARATION THEREOF H. LUNDBECK A/S (DK) 1988-05-04 EP disclosed
US-4608378-A Tetrahydroisoxazolo[4,5-c]pyridine derivatives useful in the treatment of malfunctions of the acetylcholine or muscarinic systems H. LUNDBECK A/S (DK) 1986-08-26 US disclosed