SCHEMBL10657808

SCHEMBL10657808

CCc1nc2ccc(Cl)cc2c(=O)n1CCCn1ccnc1

nearest known ligand 0.59

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.58
CYP3A4 P08684 1/20 0.58
CYP2D6 P10635 1/20 0.58
CYP2C9 P11712 1/20 0.58
CYP2C19 P33261 1/20 0.58
SMN1; SMN2 Q16637 1/20 0.58
TSHR P16473 1/20 0.54
MAPK1 P28482 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
ESR1 P03372 1/20 0.52
ALOX15 P16050 1/20 0.52
HSD17B10 Q99714 1/20 0.52
GAA P10253 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10653098 0.87 TSHR (0.72) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL15457139 0.74 KDM4E (0.50) CYP3A4TSHRMAPK1ALOX15GAA
SCHEMBL10736548 0.73
SCHEMBL10757805 0.73
SCHEMBL10654289 0.73
SCHEMBL3232811 0.73 MAPT (0.46) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL10660769 0.73
SCHEMBL10654564 0.73
SCHEMBL10659233 0.73
SCHEMBL10733601 0.73

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0293500-A1 3-heteroalkyl-2,4.quinzaoline-diones AMERICAN CYANAMID COMPANY (US) 1988-12-07 EP disclosed
US-4753944-A INHIBITING THROMBOXANE SYNTHETASE AMERICAN CYANAMID COMPANY (US) 1988-06-28 US disclosed
US-4710502-A THROMBOXANE SYNTHETASE INHIBITORS AMERICAN CYANAMID COMPANY (US) 1987-12-01 US disclosed