SCHEMBL10672014

SCHEMBL10672014

NCCCOc1cccc(CCN2CCCCC2)c1

nearest known ligand 0.62

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 5/20 0.62
KCNH2 Q12809 2/20 0.61
KDM4E B2RXH2 2/20 0.59
ALDH1A1 P00352 2/20 0.59
SMN1; SMN2 Q16637 1/20 0.59
L3MBTL1 Q9Y468 1/20 0.56
TSHR P16473 1/20 0.54
SIGMAR1 Q99720 1/20 0.54
BACE1 P56817 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4386868 0.88 KDM4E (0.60) HRH3KCNH2KDM4EALDH1A1SMN1; SMN2
SCHEMBL26985810 0.86 KDM4E (0.70) HRH3KCNH2KDM4EALDH1A1SMN1; SMN2
SCHEMBL30831555 0.86 KDM4E (0.70) HRH3KCNH2KDM4EALDH1A1SMN1; SMN2
SCHEMBL10689006 0.86 HRH2 (0.61) HRH3
SCHEMBL5288663 0.86 HRH2 (0.61) HRH3
SCHEMBL10679839 0.86 HRH2 (0.61) HRH3
SCHEMBL30597717 0.86 HRH2 (0.61) HRH3
SCHEMBL10527698 0.86 HRH2 (0.61) HRH3
SCHEMBL9551700 0.85 HRH2 (0.59) HRH3KDM4EALDH1A1SMN1; SMN2
SCHEMBL9574750 0.82 HRH2 (0.61) HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4738969-A Substituted aminopyridones and aminoquinolones having histamine H2 -receptor blocking activity SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1988-04-19 US disclosed
US-4608380-A HISTAMINE H2-ANTAGONISTS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1986-08-26 US disclosed