SCHEMBL10691404

SCHEMBL10691404

Nc1cc2cc(Cl)c(Cl)cc2cc1N

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.50
CD44 P16070 1/20 0.46
PTK2 Q05397 1/20 0.44
TSHR P16473 6/20 0.41
CYP3A4 P08684 6/20 0.41
ALDH1A1 P00352 3/20 0.41
ALOX15 P16050 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
AHR P35869 2/20 0.40
FLT1 P17948 1/20 0.40
TP53 P04637 1/20 0.39
MAPK1 P28482 2/20 0.38
CASP6 P55212 1/20 0.37
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
CA14 Q9ULX7 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26746409 0.87 GAA (0.69) GAACD44PTK2TSHRCYP3A4
SCHEMBL203217 0.82 GAA (0.71) GAACD44PTK2TSHRCYP3A4
SCHEMBL29534050 0.82 GAA (0.71) GAACD44PTK2TSHRCYP3A4
SCHEMBL5792991 0.82 AHR (0.47) GAATSHRCYP3A4ALDH1A1SMN1; SMN2
SCHEMBL29429002 0.82 PTK2 (0.64) GAACD44PTK2TSHRCYP3A4
SCHEMBL1599775 0.82 PTK2 (0.64) GAACD44PTK2TSHRCYP3A4
SCHEMBL11251343 0.81 HSD17B10 (0.44) GAATSHRCYP3A4ALDH1A1ALOX15
Ammonia Solution, Strong SCHEMBL8321418 0.79 GAA (0.67) GAACD44PTK2TSHRCYP3A4
SCHEMBL27937186 0.79 GAA (0.67) GAACD44PTK2TSHRCYP3A4
Ammonia Solution, Strong SCHEMBL7755770 0.79 GAA (0.67) GAACD44PTK2TSHRCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4792508-A STEREOISOMERIC NAPHTHALENE IMIDAZOLE PERYLENES, ARYL AMINES XEROX CORPORATION (US) 1988-12-20 US disclosed
EP-0042753-B1 NONAPEPTIDE AND DECAPEPTIDE AGONISTS OF LUTEINIZING HORMONE RELEASING HORMONE CONTAINING HETEROCYCLIC AMINO ACID RESIDUES, METHODS FOR THEIR PREPARATION, PHARMACEUTICAL COMPOUNDS CONTAINING THEM, AND THEIR PHARMACEUTICAL USE SYNTEX (U.S.A.) INC. (US) 1984-03-21 EP disclosed
US-4318905-A Nonapeptide and decapeptide agonists of luteinizing hormone releasing hormone containing heterocyclic amino acid residues SYNTEX (U.S.A.) INC. (US) 1982-03-09 US disclosed
EP-0042753-A1 Nonapeptide and decapeptide agonists of luteinizing hormone releasing hormone containing heterocyclic amino acid residues, methods for their preparation, pharmaceutical compounds containing them, and their pharmaceutical use SYNTEX (U.S.A.) INC. (US) 1981-12-30 EP disclosed