SCHEMBL10695086

SCHEMBL10695086

CN1C(=O)C(C)(C)c2cc3c(cc21)nc(-c1ccc(O)cc1)n3C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
PDE4A P27815 2/20 0.39
PDE4B Q07343 2/20 0.39
PDE4C Q08493 2/20 0.39
PDE4D Q08499 2/20 0.39
PKM P14618 3/20 0.38
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
CNR1 P21554 1/20 0.38
GPR55 Q9Y2T6 1/20 0.38
HDAC1 Q13547 2/20 0.37
HDAC8 Q9BY41 2/20 0.37
HDAC6 Q9UBN7 2/20 0.37
ESR1 P03372 1/20 0.36
JAK2 O60674 1/20 0.36
JAK1 P23458 1/20 0.36
TYK2 P29597 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10697084 0.95 MEN1 (0.40) MEN1KMT2APDE4APDE4BPDE4C
SCHEMBL10695690 0.87 MEN1 (0.47) MEN1KMT2APDE4APDE4BPDE4C
SCHEMBL10698656 0.86 BRD4 (0.46) MEN1KMT2APKMCA12CA1
SCHEMBL10700878 0.86 POLB (0.40) MEN1KMT2APDE4APDE4BPDE4C
SCHEMBL10709508 0.85 DHODH (0.41) MEN1KMT2APKMCA12CA1
SCHEMBL10697337 0.84 BRD4 (0.37) MEN1KMT2ACA12CA1CA2
SCHEMBL10695172 0.82 MEN1 (0.47) MEN1KMT2APDE4APDE4BPDE4C
SCHEMBL10697806 0.82 BRD4 (0.50) MEN1KMT2APKMCA12CA1
SCHEMBL10700736 0.81 BRD4 (0.41) MEN1KMT2APKMCA12CA1
SCHEMBL10698013 0.77 CA12 (0.50) MEN1KMT2APDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0268178-A1 Pyrrolo-benzimidazoles, medicaments containing these compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1988-05-25 EP disclosed