SCHEMBL10697812

SCHEMBL10697812

O=C(O)[C@H](Br)CCc1ccc([N+](=O)[O-])cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.54
ANPEP P15144 1/20 0.48
ERAP2 Q6P179 1/20 0.48
ERAP1 Q9NZ08 1/20 0.48
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
CYP2C19 P33261 2/20 0.45
CYP1A2 P05177 1/20 0.45
KCNH2 Q12809 2/20 0.45
KCNJ1 P48048 1/20 0.45
MAPT P10636 2/20 0.45
LOXL2 Q9Y4K0 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
TAAR1 Q96RJ0 1/20 0.44
ALDH1A1 P00352 2/20 0.44
GSK3B P49841 1/20 0.44
PTGES O14684 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27311205 1.00 TSHR (0.54) TSHRANPEPERAP2ERAP1MEN1
SCHEMBL4373315 1.00 TSHR (0.54) TSHRANPEPERAP2ERAP1MEN1
SCHEMBL3097653 0.86 TSHR (0.61) TSHRANPEPERAP2ERAP1MEN1
SCHEMBL2438048 0.83 MEN1 (0.49) TSHRANPEPERAP2ERAP1MEN1
SCHEMBL2561037 0.82 TSHR (0.56) TSHRANPEPERAP2ERAP1MEN1
SCHEMBL2603379 0.82 TSHR (0.49) TSHRMEN1KMT2AKCNH2KCNJ1
SCHEMBL10610015 0.81 MAPT (0.51) TSHRMEN1KMT2AKCNH2KCNJ1
SCHEMBL10610005 0.81 MAPT (0.51) TSHRMEN1KMT2AKCNH2KCNJ1
SCHEMBL10610012 0.81 MAPT (0.51) TSHRMEN1KMT2AKCNH2KCNJ1
SCHEMBL8092467 0.81 GRM8 (0.56) TSHRANPEPERAP2ERAP1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0271795-A2 Octahydro-10-oxo-6H-pyridazo[1,2-a][1,2]diazepin derivatives, intermediates and process for their preparation, and medicament containing them F. HOFFMANN-LA ROCHE AG (CH) 1988-06-22 EP disclosed