SCHEMBL1070276

SCHEMBL1070276

C=CCN1C(=O)[C@@](C)(CF)N(C)CC1(C)c1cc(F)cc(F)c1

nearest known ligand 0.38

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CALCRL Q16602 10/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL979348 1.00 CALCRL (0.38) CALCRLPTGDR2
SCHEMBL979347 1.00 CALCRL (0.38) CALCRLPTGDR2
SCHEMBL979128 1.00 CALCRL (0.38) CALCRLPTGDR2
SCHEMBL979126 1.00 CALCRL (0.38) CALCRLPTGDR2
SCHEMBL979129 1.00 CALCRL (0.38) CALCRLPTGDR2
SCHEMBL976466 0.89 CALCRL (0.37) CALCRLPTGDR2
SCHEMBL976469 0.89 CALCRL (0.37) CALCRLPTGDR2
SCHEMBL980013 0.81 CALCRL (0.35) CALCRL
SCHEMBL980014 0.81 CALCRL (0.35) CALCRL
SCHEMBL980015 0.81 CALCRL (0.35) CALCRL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2271346-A2 MONOCYCLIC CGRP RECEPTOR ANTAGONISTS Merck Sharp & Dohme Corp. (US) 2011-01-12 EP disclosed
WO-2009120652-A2 MONOCYCLIC CGRP RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2009-10-01 WO disclosed