SCHEMBL1072809

SCHEMBL1072809

O=C(NC[C@@H]1CCCO1)c1ccc(C(=O)N(Cl)c2ccc(Cl)c(-c3ccccn3)c2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 3/20 0.54
MAPT P10636 1/20 0.54
HPGD P15428 6/20 0.53
SMN1; SMN2 Q16637 3/20 0.52
KMT2A Q03164 2/20 0.52
NPC1 O15118 2/20 0.52
MEN1 O00255 1/20 0.51
CYP2C9 P11712 2/20 0.49
ALDH1A1 P00352 4/20 0.48
TSHR P16473 2/20 0.48
KDM4E B2RXH2 1/20 0.48
TP53 P04637 1/20 0.48
HSD17B10 Q99714 1/20 0.48
ATM Q13315 1/20 0.48
RAB9A P51151 2/20 0.47
CYP1A2 P05177 1/20 0.46
GAA P10253 1/20 0.46
CYP2C19 P33261 1/20 0.46
GLA P06280 1/20 0.46
ALOX12 P18054 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1253725 0.80 ATM (0.55) POLBMAPTHPGDSMN1; SMN2CYP2C9
SCHEMBL30572146 0.80 ATM (0.55) POLBMAPTHPGDSMN1; SMN2CYP2C9
SCHEMBL1018147 0.79 ATM (0.54) POLBMAPTHPGDSMN1; SMN2ALDH1A1
SCHEMBL14082186 0.79 HPGD (0.71) POLBMAPTHPGDSMN1; SMN2KMT2A
SCHEMBL1071329 0.78 NTRK1 (0.47) HPGD
SCHEMBL2119183 0.74 KDM4E (0.44) POLBMAPTSMN1; SMN2ALDH1A1KDM4E
SCHEMBL30865898 0.74 KDM4E (0.44) POLBMAPTSMN1; SMN2ALDH1A1KDM4E
SCHEMBL26036542 0.74 NAMPT (0.42) POLBMAPTSMN1; SMN2ALDH1A1KDM4E
SCHEMBL743611 0.72 HPGD (1.00) POLBHPGDSMN1; SMN2KMT2ANPC1
SCHEMBL29687327 0.72 HPGD (1.00) POLBHPGDSMN1; SMN2KMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2271642-A2 PYRIDYL INHIBITORS OF HEDGEHOG SIGNALLING Genentech, Inc. (US) 2011-01-12 EP disclosed
WO-2009126863-A2 PYRIDYL INHIBITORS OF HEDGEHOG SIGNALLING GENENTECH, INC. (US) 2009-10-15 WO disclosed