SCHEMBL10739945

SCHEMBL10739945

NC1CCCC/C1=C\c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.44
MAPT P10636 2/20 0.44
CHRNB2 P17787 1/20 0.43
CHRNB4 P30926 1/20 0.43
CHRNA3 P32297 1/20 0.43
CHRNA4 P43681 1/20 0.43
CHRNA7 P36544 1/20 0.43
CYP1A2 P05177 3/20 0.40
F3 P13726 1/20 0.40
LMNA P02545 2/20 0.40
ALDH1A1 P00352 2/20 0.39
HTT P42858 1/20 0.39
POLB P06746 1/20 0.38
GAA P10253 1/20 0.38
KDM1A O60341 3/20 0.36
NOS1 P29475 2/20 0.36
NOS2 P35228 2/20 0.36
AKR1C3 P42330 1/20 0.36
CYP2D6 P10635 1/20 0.34
CYP2C19 P33261 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10734159 1.00 HPGD (0.44) HPGDMAPTCHRNB2CHRNB4CHRNA3
SCHEMBL8541864 1.00 HPGD (0.44) HPGDMAPTCHRNB2CHRNB4CHRNA3
SCHEMBL10672586 0.86 CA1 (0.40) HPGDMAPTCHRNB2CHRNB4CHRNA3
SCHEMBL10736750 0.81 MAPT (0.46) HPGDMAPTCYP1A2LMNAALDH1A1
SCHEMBL10736754 0.81 MAPT (0.46) HPGDMAPTCYP1A2LMNAALDH1A1
SCHEMBL10740869 0.81 AKR1C3 (0.37) MAPTCYP1A2KDM1AAKR1C3
SCHEMBL10740873 0.81 AKR1C3 (0.37) MAPTCYP1A2KDM1AAKR1C3
SCHEMBL15987564 0.79 HPGD (0.42) HPGDMAPTCHRNB2CHRNB4CHRNA3
SCHEMBL15987566 0.79 HPGD (0.42) HPGDMAPTCHRNB2CHRNB4CHRNA3
SCHEMBL10743401 0.79 HPGD (0.41) HPGDKDM1AAKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4652559-A ANALGESIC, ANTIDEPRESSANT THE UPJOHN COMPANY (US) 1987-03-24 US disclosed
EP-0085811-B1 2-(PHENYLMETHYLENE)CYCLOALKYLAMINES THE UPJOHN COMPANY (US) 1986-05-07 EP disclosed
US-4540690-A ANALGESICS, ANTIDEPRESSANTS THE UPJOHN COMPANY (US) 1985-09-10 US disclosed
EP-0085811-A1 2-(Phenylmethylene)cycloalkylamines THE UPJOHN COMPANY (US) 1983-08-17 EP disclosed