SCHEMBL10744191

SCHEMBL10744191

COC(=O)C1=C(C)NC(C)=C(C(=O)OCCC=Cc2ccccc2)C1c1cccc([N+](=O)[O-])c1

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 6/20 0.78
KMT2A Q03164 6/20 0.78
ADORA3 P0DMS8 4/20 0.78
CACNA1C Q13936 3/20 0.78
CACNA1B Q00975 2/20 0.78
TBXA2R P21731 2/20 0.78
HTT P42858 2/20 0.78
MLNR O43193 1/20 0.78
NR1I2 O75469 1/20 0.78
CACNA1H O95180 1/20 0.78
NR3C1 P04150 1/20 0.78
PDE4D Q08499 1/20 0.78
SLC29A1 Q99808 1/20 0.78
MAPT P10636 7/20 0.71
CYP1A2 P05177 6/20 0.71
CYP3A4 P08684 6/20 0.71
CYP2C9 P11712 6/20 0.71
CYP2C19 P33261 6/20 0.71
CYP2D6 P10635 5/20 0.71
HIF1A Q16665 4/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10744188 1.00 MEN1 (0.78) MEN1KMT2AADORA3CACNA1CCACNA1B
SCHEMBL10745195 0.95 CACNA1C (0.75) MEN1KMT2AADORA3CACNA1CCACNA1B
SCHEMBL10745200 0.95 CACNA1C (0.75) MEN1KMT2AADORA3CACNA1CCACNA1B
SCHEMBL9835079 0.95 MEN1 (0.71) MEN1KMT2AADORA3CACNA1CCACNA1B
SCHEMBL9835087 0.95 MEN1 (0.71) MEN1KMT2AADORA3CACNA1CCACNA1B
SCHEMBL9831212 0.94 MEN1 (0.70) MEN1KMT2AADORA3CACNA1CCACNA1B
SCHEMBL9831217 0.94 MEN1 (0.70) MEN1KMT2AADORA3CACNA1CCACNA1B
SCHEMBL9833239 0.94 CACNA1B (0.83) MEN1KMT2AADORA3CACNA1CCACNA1B
SCHEMBL10744635 0.92 MEN1 (0.68) MEN1KMT2AADORA3CACNA1CCACNA1B
SCHEMBL10744627 0.92 MEN1 (0.68) MEN1KMT2AADORA3CACNA1CCACNA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4672068-A Antihypertensive 1,4-dihydropyridines having a conjugated ester FUJIREBIO KABUSHIKI KAISHA (JP) 1987-06-09 US disclosed
EP-0161877-A2 1,4-dihydropyridine derivatives, methods for their production and pharmaceutical compositions comprising the same FUJIREBIO KABUSHIKI KAISHA also trading as FUJIREBIO INC. (JP) 1985-11-21 EP disclosed