SCHEMBL10747985

SCHEMBL10747985

Oc1ccc(-c2cn3c(n2)CNCC3)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 1/20 0.53
CD274 Q9NZQ7 1/20 0.53
MAPT P10636 2/20 0.50
TLR9 Q9NR96 1/20 0.47
TLR8 Q9NR97 1/20 0.47
TLR7 Q9NYK1 1/20 0.47
WDR5 P61964 6/20 0.44
LMNA P02545 4/20 0.44
NPC1 O15118 4/20 0.44
RAB9A P51151 4/20 0.44
HTT P42858 2/20 0.44
ALDH1A1 P00352 3/20 0.43
KDM4E B2RXH2 1/20 0.43
PTGS1 P23219 1/20 0.41
KMT2A Q03164 2/20 0.40
GAA P10253 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
HDAC2 Q92769 3/20 0.39
HDAC1 Q13547 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15933525 0.86 PDCD1 (0.52) PDCD1CD274MAPTTLR9TLR8
SCHEMBL12781800 0.86 PDCD1 (0.52) PDCD1CD274MAPTTLR9TLR8
SCHEMBL10747141 0.86 PDCD1 (0.52) PDCD1CD274MAPTTLR9TLR8
SCHEMBL10750012 0.86 PDCD1 (0.52) PDCD1CD274MAPTTLR9TLR8
SCHEMBL15933686 0.86 NPC1 (0.61) PDCD1CD274MAPTTLR9TLR8
SCHEMBL15933440 0.86 PDCD1 (0.59) PDCD1CD274MAPTTLR9TLR8
SCHEMBL108698 0.86 PDCD1 (0.69) PDCD1CD274MAPTTLR9TLR8
Hydrochloric Acid SCHEMBL19664801 0.85 PDCD1 (0.51) PDCD1CD274MAPTTLR9TLR8
SCHEMBL15933687 0.84 PDCD1 (0.53) PDCD1CD274MAPTTLR9TLR8
SCHEMBL15933693 0.84 NPC1 (0.55) PDCD1CD274MAPTTLR9TLR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4670445-A VASODILATORS ELI LILLY AND COMPANY (US) 1987-06-02 US disclosed
US-4578387-A VASODILATION; DERIVATIVES OF 2-PHENYL-5,6,7,8-TETRAHYDROIMADAZO/1,2-A/PYRAZINE ELI LILLY AND COMPANY (US) 1986-03-25 US disclosed