SCHEMBL10765397

SCHEMBL10765397

COC(=O)C1=C(CF)NC(COC(N)=O)=C(C(=O)OC(C)C)C1c1cccc(Cl)c1Cl

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 5/20 0.52
CYP3A4 P08684 5/20 0.52
CYP1A2 P05177 4/20 0.52
CYP2C19 P33261 4/20 0.52
ABCB11 O95342 4/20 0.52
TBXA2R P21731 4/20 0.52
SLC6A3 Q01959 4/20 0.52
MEN1 O00255 3/20 0.52
KMT2A Q03164 3/20 0.52
ADRA1A P35348 3/20 0.52
ADORA3 P0DMS8 3/20 0.52
OPRK1 P41145 3/20 0.52
SCN5A Q14524 3/20 0.52
NR1I2 O75469 3/20 0.52
KDM4E B2RXH2 2/20 0.52
HIF1A Q16665 2/20 0.52
HSD17B10 Q99714 2/20 0.52
ABCB1 P08183 2/20 0.52
ADRB3 P13945 2/20 0.52
CYP2D6 P10635 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Lemildipine SCHEMBL49443 0.91 CYP2C9 (0.62) CYP2C9CYP3A4CYP1A2CYP2C19ABCB11
Lemildipine SCHEMBL29801339 0.91 CYP2C9 (0.62) CYP2C9CYP3A4CYP1A2CYP2C19ABCB11
Lemildipine SCHEMBL49442 0.91 CYP2C9 (0.62) CYP2C9CYP3A4CYP1A2CYP2C19ABCB11
SCHEMBL7429254 0.86 CYP2C9 (0.64) CYP2C9CYP3A4CYP1A2CYP2C19ABCB11
SCHEMBL9133557 0.84 CYP2C9 (0.50) CYP2C9CYP3A4CYP1A2CYP2C19ABCB11
SCHEMBL7330272 0.83 CYP2C9 (0.71) CYP2C9CYP3A4CYP1A2CYP2C19ABCB11
SCHEMBL9770423 0.83 CYP2C9 (0.62) CYP2C9CYP3A4CYP1A2CYP2C19ABCB11
SCHEMBL7320951 0.83 CYP2C9 (0.62) CYP2C9CYP3A4CYP1A2CYP2C19ABCB11
SCHEMBL7328156 0.80 CYP2C9 (0.78) CYP2C9CYP3A4CYP1A2CYP2C19ABCB11
SCHEMBL7432882 0.79 CYP2C9 (0.57) CYP2C9CYP3A4CYP1A2CYP2C19ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0225175-A2 Dihydropyridine derivatives, processes for their preparation and pharmaceutical compositions thereof FISONS plc (GB) 1987-06-10 EP claimed
EP-0225175-A2 Dihydropyridine derivatives, processes for their preparation and pharmaceutical compositions thereof FISONS plc (GB) 1987-06-10 EP disclosed