SCHEMBL10772468

SCHEMBL10772468

NC(=O)CCc1cccnn1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.51
P2RX7 Q99572 1/20 0.44
CTDSP1 Q9GZU7 1/20 0.44
VNN1 O95497 3/20 0.39
CES1 P23141 1/20 0.39
CAPN1 P07384 1/20 0.37
CYP2C9 P11712 1/20 0.36
NAMPT P43490 1/20 0.36
NR4A2 P43354 1/20 0.36
GOT1 P17174 1/20 0.34
RECQL P46063 1/20 0.34
EGFR P00533 1/20 0.34
SRC P12931 1/20 0.34
TBXAS1 P24557 1/20 0.33
CHRM1 P11229 1/20 0.33
HRH1 P35367 1/20 0.33
FAAH O00519 1/20 0.33
MPO P05164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30421162 1.00 CYP1A2 (0.51) CYP1A2P2RX7CTDSP1VNN1CES1
SCHEMBL2436110 0.91 CYP1A2 (0.50) CYP1A2P2RX7CTDSP1VNN1CES1
SCHEMBL27883898 0.85 CYP1A2 (0.50) CYP1A2P2RX7CTDSP1VNN1CES1
SCHEMBL31080880 0.83 CYP1A2 (0.53) CYP1A2P2RX7CTDSP1VNN1CES1
SCHEMBL25660463 0.83 CYP1A2 (0.53) CYP1A2P2RX7CTDSP1VNN1CES1
SCHEMBL30421462 0.81 CYP1A2 (0.54) CYP1A2P2RX7CTDSP1VNN1CES1
SCHEMBL12530365 0.79 CTDSP1 (0.49) CYP1A2P2RX7CTDSP1VNN1CES1
SCHEMBL3079246 0.77 CYP1A2 (0.47) CYP1A2P2RX7CTDSP1VNN1CES1
SCHEMBL21132517 0.76 RECQL (0.51) CYP1A2P2RX7CTDSP1VNN1CYP2C9
SCHEMBL6046250 0.76 CYP1A2 (0.50) CYP1A2CTDSP1VNN1CES1TBXAS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0223974-A1 N-Substituted-N-[3-(1,2,4-triazolo[4,3-b]pyridazin-6-yl)-phenyl]alkanamides, carbamates and ureas AMERICAN CYANAMID COMPANY (US) 1987-06-03 EP disclosed