SCHEMBL10806366

SCHEMBL10806366

CCCCCCCCCCCC(=O)CCCC[C@@H]1Cc2cc(O)ccc2C2CC[C@@]3(C)C(CC[C@@H]3O)C21

nearest known ligand 0.81

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 10/20 0.81
ESR2 Q92731 5/20 0.81
HDAC3 O15379 2/20 0.78
HDAC6 Q9UBN7 1/20 0.78
ESRRA P11474 9/20 0.64
CYP3A4 P08684 2/20 0.64
CYP2C19 P33261 2/20 0.64
NR1I2 O75469 1/20 0.64
NR3C1 P04150 1/20 0.64
PGR P06401 1/20 0.64
EPHX2 P34913 1/20 0.64
PPARG P37231 1/20 0.64
NR1H4 Q96RI1 1/20 0.64
SIRT5 Q9NXA8 1/20 0.64
CYP1A2 P05177 1/20 0.64
ALOX15 P16050 1/20 0.64
ESRRB O95718 8/20 0.59
CYP2C8 P10632 1/20 0.53
CYP2D6 P10635 1/20 0.53
CYP2C9 P11712 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10806360 1.00 ESR1 (0.81) ESR1ESR2HDAC3HDAC6ESRRA
SCHEMBL10800287 0.98 ESR1 (0.81) ESR1ESR2HDAC3HDAC6ESRRA
SCHEMBL10800292 0.98 ESR1 (0.81) ESR1ESR2HDAC3HDAC6ESRRA
SCHEMBL14094329 0.94 ESR1 (0.79) ESR1ESR2HDAC3HDAC6ESRRA
SCHEMBL26158824 0.94 ESR1 (0.79) ESR1ESR2HDAC3HDAC6ESRRA
SCHEMBL13139941 0.94 ESR1 (0.79) ESR1ESR2HDAC3HDAC6ESRRA
SCHEMBL10807820 0.91 ESR1 (0.95) ESR1ESR2HDAC3HDAC6ESRRA
SCHEMBL10972000 0.91 ESR1 (0.95) ESR1ESR2HDAC3HDAC6ESRRA
SCHEMBL10971997 0.91 ESR1 (0.95) ESR1ESR2HDAC3HDAC6ESRRA
SCHEMBL10807827 0.91 ESR1 (0.95) ESR1ESR2HDAC3HDAC6ESRRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4659516-A ANTIESTROGENS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1987-04-21 US disclosed
EP-0138504-A2 Steroid derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1985-04-24 EP disclosed